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5-ethyl-N-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-(4-ethyl-1H-pyrazol-5-yl)-1-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]piperidine
5-{3-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
1-(butan-2-yl)-N3-ethyl-N5-[2-(1H-indol-3-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(2-methoxyacetyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
1-[2-(4-fluorophenoxy)pyridin-3-yl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
5-(hydroxymethyl)-4-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2-methylpyridin-3-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2,3-trimethylbenzamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentane-1,4-dione
N-[2-(4-fluorobenzenesulfonyl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
4-benzyl-3-ethyl-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
1-(benzenesulfonyl)-3-(3-chlorobenzoyl)piperidine
3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}benzoic acid
N-[3-(dimethylamino)propyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
9-(2-ethylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-5-(2-oxo-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{imidazo[1,2-a]pyridin-2-yl}-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
N-{1-[1-(3-hydroxy-2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,4-dihydroquinolin-4-one
(2S,3R)-3-hydroxy-2-{4-[2-(piperidin-1-yl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}butanoic acid
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(6-methoxypyrimidin-4-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-(1-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(3-methylpyridin-2-yl)ethyl]pyridin-2-amine
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine-2-carboxamide
1-[(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(trifluoromethyl)benzamide
1-(5-chloro-2-ethoxy-4-methylbenzenesulfonyl)-4-(hydroxymethyl)azepan-4-ol
[2-(2,4-dimethylphenoxy)ethyl](methyl){[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N5-tert-butyl-1-cyclohexyl-N3-(2-hydroxy-2-phenylethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(3-fluorophenyl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-(cyclohexylmethyl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-4-methoxyoxolan-3-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-3-hydroxy-2,2-dimethylpropan-1-one
1-[2-(1H-imidazol-2-yl)benzoyl]-3-(4-methylphenoxymethyl)piperidine
N-(2-methoxyethyl)-3-methyl-4-oxo-N-(pyridin-2-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
methyl 4-{4-[3-(pyridin-3-yl)propanoyl]piperazin-1-yl}benzoate
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-amino-1-{[1-(5-carboxy-2-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methyl}pyrrolidine-3-carboxylic acid
N-cyclopentyl-1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-(3-fluorophenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-methyl-2-[1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
[(3S,5R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
2-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-[2-(3-fluorophenyl)ethyl]-4-[4-(thiophen-3-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione