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[(5-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
7,7-dimethyl-2-{6-methylimidazo[1,2-a]pyridin-2-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-3-methyl-1-[2-(propylsulfanyl)phenyl]urea
9-(cyclopropylmethyl)-1-methyl-4-(pyrazin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[3-(4-hydroxypiperidin-1-yl)-3-oxopropyl]-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-chloro-N-(3-hydroxypropyl)-3-methyl-N-(thiophen-2-ylmethyl)-1H-indole-2-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
{1-[4-(4-{[(2-methoxynaphthalen-1-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
N-[2-(pyrrolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-{1-[1-(2-ethoxyethyl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-N-methylacetamide
N-(1-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1-ethylpiperidine-4-carboxamide
N-[(3S,4R)-1-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
(1S,5R)-6-(cyclopropylmethyl)-N-(2-methoxy-5-methylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-cyclohexyl-4-(3-hydroxypyridine-2-carbonyl)piperazin-2-one
N-benzyl-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-5-methyl-1-propyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-(1-butyl-5-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}-1H-1,2,4-triazol-3-yl)acetamide
2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]pyridine-3-carbonitrile
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(hydroxymethyl)quinolin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethylpiperidin-4-amine
1-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
5-[benzyl(methyl)amino]-2-(2-hydroxybutyl)-2,3-dihydropyridazin-3-one
3-[2-(4-fluorophenyl)ethyl]-1-(1H-imidazol-4-ylmethyl)piperidine
1-{4-[(6-ethyl-4-methylquinolin-2-yl)amino]piperidin-1-yl}-2-methylpropan-1-one
2-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-6-methylpyridine
3-chloro-6-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
1-(2-{4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-cyclopentyl-4-(3-hydroxybenzoyl)piperazin-2-one
(5S)-5-({[(1-ethyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amino}methyl)pyrrolidin-2-one
N-cyclopentyl-1-(4,7-dimethylquinazolin-2-yl)azepan-4-amine
3-{5-cyclopentyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
3-{[(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
N-[(1-ethylpyrrolidin-3-yl)methyl]-5-methyl-2,1,3-benzothiadiazole-4-sulfonamide
methyl 1-ethyl-3-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)-1H-pyrrolo[2,3-c]pyridine-5-carboxylate
3-(2-amino-1,3-thiazol-4-yl)-N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]propanamide
7-hydroxy-4-(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
2-ethyl-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)pyrimidine-5-carboxamide
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
4-[3-(benzyloxy)propyl]-N,N-dimethylbenzamide
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-methyl-3-(2-methylpropyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
(1R,5R)-6-[2-(benzyloxy)ethyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(3S,4S)-1-[(5-tert-butyl-2-hydroxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-(1-cycloheptylpiperidin-3-yl)-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide