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9-methyl-3-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
[(4aS,8aR)-6-[(2,3-difluoro-6-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
N-[3-(2-oxopyrrolidin-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(4S)-1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
1-methyl-3-phenyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
N-[3-(pyridin-2-yl)propyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-(4-methoxyphenoxymethyl)-N-(2-oxopyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(2-methoxyphenoxy)piperidine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}-1,2,3-thiadiazole-4-carboxamide
N-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]-1-azabicyclo[2.2.2]octan-3-amine
[(1R,3S,3aS,6aR)-3-(1,5-dimethyl-1H-pyrazol-4-yl)-5-ethyl-1-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(2R,3R,6R)-5-(2-chlorobenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methyl-3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
6-[methyl(pyrazin-2-ylmethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N,N-dimethyl-2-[4-(1-{3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl}-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide
N-(1-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)acetamide
(1S,5R)-6-(pyrrolidine-1-sulfonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(2-phenylethyl)piperidine-4-carboxamide
3-{1-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperidin-4-yl}propanoic acid
5-[4-(ethylsulfanyl)phenyl]pyrazin-2-amine
5-{[1-cyclohexyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
(4aS,8aR)-1-butyl-6-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-(4-acetylphenyl)-3-[(2-methylphenyl)methyl]-3-(oxolan-2-ylmethyl)urea
2-(3,3-diphenylpiperidin-1-yl)-1-(morpholin-4-yl)ethan-1-one
2-methyl-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,3-thiazole-4-carboxamide
2,2-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}oxane-4-carboxamide
5-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
1-[(3,5-dichloro-2-methoxyphenyl)methyl]-3-methoxypyrrolidine
N-[2-(3-methoxyphenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(phenylsulfanyl)acetamide
(3S,9aR)-3-(propan-2-yl)-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[2-(benzyloxy)phenyl]-3-[(1-ethylpyrrolidin-2-yl)methyl]urea
(1R,5S,6S)-6-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
2-(2,3-dihydro-1H-inden-2-yl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(ethanesulfonyl)-4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
2-methoxy-1-{1'-[(6-methylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(4aR,7aS)-1-butanoyl-4-[3-(thiophen-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
1-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-(2-fluoro-6-methoxybenzoyl)-4-(1-methylpiperidin-4-yl)piperazine
6-methyl-2-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
6-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-4-methyl-1,3-benzothiazol-2-amine
2-methyl-8-[2-(methylamino)pyridine-3-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine