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2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1,4-dihydroquinolin-4-one
3,3-dimethyl-1-({5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
5-(2-chloro-4-methoxyphenoxymethyl)-N-(pentan-2-yl)-1H-pyrazole-3-carboxamide
ethyl 1-(2-methylfuran-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}pyridine
(1s,4s)-4-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}cyclohexan-1-amine
1-benzyl-5-{[(5-chlorothiophen-2-yl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl}benzoic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-4,4,4-trifluorobutanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
2-[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)amino]-N,N-dimethylpropanamide
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
methyl (2S,4S)-1-[(2,6-difluorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
2-{3-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxymethyl}pyridine
N-{2-[(3S,4R)-3-cyclopropyl-4-[(2-methylpyrimidin-4-yl)amino]pyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-phenylbutane-1,2-dione
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-propyl-1,2,3-thiadiazole-5-carboxamide
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-5-{1-[2-(methylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-cyclopentyl-9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-hydroxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(3-methylphenyl)pyrimidine-5-carboxamide
3-ethyl-8-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-methoxy-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
N-cyclopropyl-1-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperazine-2-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-cyclopentyl-5-oxo-N-[2-(1,3-thiazol-4-yl)ethyl]pyrrolidine-3-carboxamide
4-({[cyclopropyl(4-methylpyridin-2-yl)methyl]carbamoyl}amino)-N-ethyl-3-methylbenzamide
N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
6-methoxy-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
1-[3-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidin-4-ol
3-(3-methoxyphenoxymethyl)-1-(thiophene-3-carbonyl)piperidine
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
4-[1-(1-cycloheptanecarbonylpiperidin-4-yl)piperidine-4-carbonyl]morpholine
3-{2-[(7-fluoroquinazolin-4-yl)amino]ethyl}-4-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2-fluorophenyl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-2-(2-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
ethyl 2-(1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)acetate
N-[(2S,3S)-1-hydroxy-3-methylpentan-2-yl]-2,6-dimethylpyridine-4-carboxamide
(2S,4S)-4-[4-({[(3-chloro-2-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
(3S,4R)-1-(4-chloro-3-methylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
(2S)-3-methyl-2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]butanamide
(2S,4S)-4-amino-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
[(1-benzyl-1H-pyrazol-4-yl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-(2-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
2-(2-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
3-{[3-(ethoxymethyl)-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1H-isoindol-1-one