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N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(pyridin-2-yl)acetamide
ethyl 4-(2-phenylethyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-4-carboxylate
8-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-[3-chloro-2-(propan-2-yloxy)phenyl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
N-tert-butyl-2-[(4-fluorophenyl)methyl]morpholine-4-carboxamide
dimethyl({4-methyl-5-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2,6-dimethoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-4-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]methylamine
N-[(3S,4R)-1-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
methyl 2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-oxopiperazin-2-yl}acetate
N-[4-(pyridin-3-yloxy)phenyl]-1-[(2R)-pyrrolidine-2-carbonyl]piperidine-4-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
(1R,2S)-2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N-methylcyclohexane-1-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
N4-methyl-6-(4-methylpiperazin-1-yl)-N4-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine
4-(piperidine-1-carbonyl)-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
2-amino-4-[2-(cyclopentylmethyl)-1H-imidazol-4-yl]-6-ethyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-2-propyl-1,3-thiazole
3-amino-1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
(3S,4R)-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-(3-fluoro-4-methoxyphenyl)quinolin-4-amine
2-chloro-4-fluoro-N-(3-methoxy-2,2-dimethylpropyl)benzamide
6-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-methyl-4-[3-(2-methyl-1,3-thiazol-4-yl)-5-(phenoxymethyl)-1H-1,2,4-triazol-1-yl]piperidine
N-[(3S,4R)-4-(propan-2-yl)-1-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)pyrrolidin-3-yl]acetamide
N-{[1-(2,5-dichlorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,4,4-trifluorobutanamide
(3S,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[ethyl(3-methylphenyl)amino]ethyl}acetamide
3-(4-chloro-1H-pyrazol-1-yl)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)propanamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2H-1,3-benzodioxol-5-yl)acetamide
2-[3-(pyridin-4-yl)azetidin-1-yl]-1,3-thiazole-4-carboxamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl]-1H-1,2,4-triazol-1-yl}acetic acid
1-{4-[2-methoxy-5-(1,2-oxazinane-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[methyl(2-methylpropyl)carbamoyl]pyrrolidine-2-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}propan-1-one
2-(4-cyclopentyl-1,4-diazepan-1-yl)pyrimidin-4-amine
1-[(4aS,8aR)-1-[3-(benzyloxy)propyl]-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(azepan-1-yl)-2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]ethane-1,2-dione
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-1H-imidazole-5-carboxamide
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
[5-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
2-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)-3,4-dihydroquinazolin-4-one
4-chloro-2-{[3-(morpholin-4-yl)piperidin-1-yl]methyl}phenol
3-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}piperidine-1-carboxamide