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N-[2-(cyclohex-1-en-1-yl)ethyl]-5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
1-{2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]ethyl}piperidine-3-carboxamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)morpholine-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-ol
2-(2,3-dihydro-1H-inden-1-yl)-1-[6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl]ethan-1-one
5-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]acetamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-2-(pyridin-2-yl)acetamide
methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
2-(3-chlorophenyl)-4-[3-(piperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-{2-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
2-amino-6-cyclopropyl-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-ethyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
N-(4-fluorophenyl)-1-(pyridine-3-carbonyl)piperidin-3-amine
N-[(3R,4R)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
(4aS,8aS)-2-(1-benzofuran-2-ylmethyl)-decahydroisoquinolin-4a-ol
5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-(pyridin-2-yl)azetidine-1-carboxamide
2-[methyl({4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl})amino]ethan-1-ol
1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazole
2-(1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-2-yl)pyridine
1-{1-[2-(difluoromethoxy)benzoyl]piperidin-3-yl}-2-phenylethan-1-one
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
2-cyclopropyl-5-[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
1-(cyclohexylmethyl)-N-ethyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-ethyl-1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidine-3-carboxylic acid
3-[4-(1-hydroxy-3-phenylpropyl)piperidine-1-carbonyl]-2-methylphenol
[2,4,6-trimethyl-3-({[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amino}methyl)phenyl]methanol
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(2-methoxyphenyl)methyl]piperidine
1-{4-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]piperidin-1-yl}butan-1-one
4-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-5-methyl-1,3-oxazole
(4aS,7aR)-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane
ethyl(pyridin-2-ylmethyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
(3R,4S)-1-(3-chlorobenzenesulfonyl)-4-cyclopropylpyrrolidin-3-amine
2-(3-acetyl-1H-indol-1-yl)-N-(4H-1,2,4-triazol-4-yl)butanamide
8-(cyclohex-3-en-1-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-ol
2-(4-fluorophenyl)-1-{4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
(1R,5S,6S)-6-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-{3-[({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]pyridin-2-yl}piperidin-3-ol
methyl 4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
N-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}-2-methyl-1,3-thiazole-4-carboxamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
N-methyl-N-(oxan-2-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-amino-4-[(1-ethyl-5-oxopyrrolidin-3-yl)amino]quinazoline-6-carboxylic acid
3-(1-ethyl-1H-pyrazol-4-yl)-1-{[1-(2-fluorophenyl)cyclopentyl]methyl}urea