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2-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-5-fluoro-1H-1,3-benzodiazole
(2S)-2-(methylamino)-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N-cyclopropyl-1-(2-{1-[2-(4-methoxyphenyl)acetyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
dimethyl({5-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)amine
S-(2-cyclobutanecarbonyl-1,2,3,4-tetrahydroisoquinolin-6-yl)-3-hydroxybutane-1-sulfonamido
4-[(3-methoxypropyl)amino]-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
7-methoxy-1-methyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-chlorophenyl)methyl]-N-cyclopropylpyrrolidine-2-carboxamide
1'-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3S,4R)-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidine
(2S,4S)-4-amino-N-ethyl-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-[1-(piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
4-(3,6-dimethylpyrazin-2-yl)-2-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}phenol
3-(2-fluorophenyl)-N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
8-(5-acetylpyridin-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-methanesulfonylphenyl)methyl]-4-(oxan-4-yl)piperazine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
2-ethyl-4-methyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)-1,3-oxazole-5-carboxamide
2-(1,2,3,4-tetrahydroisoquinolin-2-yl)-1-(thiomorpholin-4-yl)propan-1-one
3-({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
4-methyl-3-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]sulfonyl}benzoic acid
4-({1-[4-(1H-pyrazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3,3-diphenylpiperidine
5-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]pyrazin-2-ol
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(5-chlorothiophen-2-yl)pyridine-3-carbonitrile
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidine-2-carboxylate
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-[(1-benzyl-1H-imidazol-5-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
N-benzyl-3-(dimethyl-1,2-oxazol-4-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]propanamide
5-methoxy-2-[4-(2-phenylethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
5-(methoxymethyl)-N-({3-methyl-7-[2-(1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
N-(4-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenyl)acetamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-N-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
4-(2,4-dimethylpyrimidine-5-carbonyl)-2-(trifluoromethyl)morpholine
6-(2-chlorophenyl)-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(1S,5R)-6-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]-3-methylpiperazin-2-one
(3S,4R)-1-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
(4aR,8aS)-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine
2-(3-hydroxyphenyl)-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
5-({2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazol-5-yl}formamido)pentanoic acid
[(3R,4R)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(5-{[(1H-indazol-6-yl)amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
4-cyano-N-(3-cyclopentaneamidophenyl)piperidine-1-carboxamide
3-methoxy-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]propanamide