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(3aR,6aS)-5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclobutanecarbonyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
2-(4-chlorophenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
(4aS,7aR)-1-[2-(4-fluoro-3-methylphenyl)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(pyrazin-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[4-(1H-indol-2-yl)phenyl]-1-(thian-4-yl)piperidine-4-carboxamide
N-cyclopropyl-7-(2,3-dihydro-1-benzofuran-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
methyl 5-[3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-5-oxopentanoate
(2S,4S)-4-amino-N,N-diethyl-1-[(5-methylthiophen-2-yl)sulfonyl]pyrrolidine-2-carboxamide
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-1,4-dioxane-2-carboxamide
(1R,2R,6S,7S)-4-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-azatricyclo[5.2.1.02,6]decane
N-[(2-fluorophenyl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[(3E)-hex-3-enoyl]pyrrolidine-3-carboxylic acid
8-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-(4-{4-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]piperidin-1-yl}benzoyl)piperidin-3-ol
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
(2R)-2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-2-phenylethan-1-ol
(3S,4S)-1-(oxan-4-yl)-4-[4-(pyridin-4-yl)piperazin-1-yl]pyrrolidin-3-ol
4-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}benzene-1-sulfonamide
(2S)-2-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]amino}-3,3-dimethylbutan-1-ol
methyl 4-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]butanoate
1-[(4-fluorophenyl)methyl]-4-[2-methyl-2-(morpholin-4-yl)propyl]-1,4-diazepane
(3R,4R)-1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
[5-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
2-[(dimethylcarbamoyl)amino]-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
3-(5-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-{2-[3-methoxy-5-(trifluoromethyl)phenyl]pyridine-4-carbonyl}-4-methylpiperazine
2-benzyl-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecane
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-(4-methoxyphenyl)-4-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperazin-2-one
8-methoxy-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-fluoroethyl)-3-methoxybenzamide
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(pyridin-3-yl)morpholine
N-cyclopropyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-propyl-1,2-oxazole-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(4aS,7aR)-1-(1-methyl-1H-pyrazole-4-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperazin-1-yl]quinazoline
4-[(6-methylpyridin-3-yl)oxy]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylic acid
3-{[4-(8-methylquinolin-5-yl)-1H-1,2,3-triazol-1-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-ethyl-1H-pyrazole
7-cyclohexyl-2-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
6-fluoro-N-(furan-2-ylmethyl)-N-methyl-1H-1,3-benzodiazole-2-carboxamide
2-[(4aR,7aS)-4-(1H-imidazol-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(methylsulfanyl)ethyl]benzamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
1-[1'-(2,4-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one