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1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
5-{2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}pyridine-2-carbonitrile
2-butyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-oxa-9-azaspiro[5.5]undecane
1-(1-benzylpiperidin-4-yl)-3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)urea
(2E)-3-(2-chlorophenyl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
5-ethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-4-(thiophene-2-carbonyl)piperazine
5-(1-ethyl-1H-imidazol-2-yl)-1-[3-(oxolan-3-yl)propyl]-4-phenyl-1H-imidazole
N-(furan-2-ylmethyl)-5-methyl-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
methyl 5-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-methyl-8-[3-(1H-pyrrol-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4,4-difluoropiperidine
4-[4-(2-fluorophenoxy)piperidin-1-yl]pyrimidine-5-carboxylic acid
2-methyl-N-{2-oxo-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}propanamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-[(2-methoxyphenyl)methyl]-4,6-dimethyl-2-oxo-N-propyl-2H-pyran-5-carboxamide
3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
N-benzyl-N-butyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
6-[1-ethyl-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
1-(3-chlorophenyl)-4-[4-(pyrrolidin-1-yl)butanoyl]piperazin-2-one
N-ethyl-N-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}oxan-4-amine
N-{[6-(4-phenoxyphenyl)pyridin-3-yl]methyl}acetamide
4-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methylfuran-2-yl)methyl]benzamide
1-(2-methyloxane-2-carbonyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
5-hydroxy-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)pyrazine-2-carboxamide
ethyl 1-[4-(4-fluorophenyl)-4-oxobutanoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
2-{[(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(1S,6R)-9-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
methyl 1-{2-hydroxy-3-[4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
3-(furan-2-yl)-5-[(6-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-amino-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
ethyl 1-(1-{[2-oxo-1-(prop-2-en-1-yl)-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidin-4-yl)piperidine-3-carboxylate
2-[5-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(4-chlorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl({[5-(pyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
(3R,5R)-1-(2-phenylethyl)-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine
1-[(1-methyl-1H-indol-3-yl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-chloro-N-(2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}ethyl)benzamide
1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(piperidin-4-ylmethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
methyl 3-[(2,2-dimethylpropanamido)methyl]-5-(thiophene-2-sulfonamido)benzoate
5-[3-(morpholin-4-ylmethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
ethyl 2-[3-(thiophene-2-carbonyl)piperidin-1-yl]acetate