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2,2,2-trifluoro-1-[4-(trimethylpyrimidin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclopropyl-1-[1-(1H-indole-6-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-[methyl({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]-1-phenylethan-1-ol
5-(1-benzofuran-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
3-{[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}benzonitrile
2-{[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]methyl}-5,8-dimethylquinolin-4-ol
N-phenyl-5-(1,3-thiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(1S,5R)-3-(pyridin-2-ylmethyl)-6-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
6-methyl-2-[(2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
2-[3-(1H-indol-3-yl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-(morpholine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(dimethylamino)phenyl]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
5-cyclopentyl-3-{[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
[(3R,4R)-1-benzoyl-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
6-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-2-methyl-1,3-benzoxazole
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(1H-imidazol-4-yl)ethyl]pyrimidin-2-amine
5-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(2-{4-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
N-cyclopropyl-3-{5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-(2-methoxyethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-(6-methylpyridazin-3-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-methoxy-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
2-{[6-(propan-2-yl)pyrimidin-4-yl]amino}-1-(pyrrolidin-1-yl)ethan-1-one
1-[2-(methylsulfanyl)pyridine-3-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[(3R,4S)-4-(dimethylamino)-1-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}piperidin-3-yl]propan-1-ol
6-methyl-2-[(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
(2S,4R)-N-ethyl-1-(1H-imidazol-2-ylmethyl)-4-[2-(propan-2-yloxy)acetamido]pyrrolidine-2-carboxamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(morpholin-4-yl)-N-(propan-2-yl)benzamide
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}-1,4-diazepan-5-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[(1r,4r)-4-hydroxycyclohexyl]-1,3-oxazole-4-carboxamide
2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1-propylpyrrolidin-2-one
3-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
(3S,4R)-N,N-dimethyl-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidin-3-amine
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-4-yl)propan-1-one
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(2-ethoxyphenyl)methyl](2-methoxyethyl)amine
3-[5-(6-chloro-8-methylquinolin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperazine
6-methyl-3-(oxan-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(pyridin-3-yloxy)propyl]acetamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[2-(2,4-difluorophenyl)-1-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
8-pentanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(4-fluorophenoxymethyl)-N-[2-(methylsulfamoyl)ethyl]-1,3-oxazole-4-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)benzamide