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(2R)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-hydroxypropanamide
2-(4-methyl-1H-pyrazol-1-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
3-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]pyridin-2-ol
N-(3,4-difluorophenyl)-1-(4-ethenylbenzoyl)piperidin-3-amine
5-methanesulfonyl-1'-(pyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
6-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoxaline
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2-(morpholin-3-yl)acetamide
(1S,5R)-3-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-2,6-dimethylphenol
2-{3-[1-(3-hydroxypropyl)-1H-pyrazol-3-yl]phenyl}-N,N-dimethylpyridine-3-carboxamide
N-(2-ethoxyphenyl)-3-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]propanamide
2-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1-(morpholin-4-yl)ethan-1-one
1-[1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(1S,5R)-3-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,5R)-N5-(2,3-dihydro-1H-inden-5-yl)-N3,N3-dimethylpiperidine-3,5-dicarboxamide
5-({4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)-2-phenylpyrimidine
2-(2-chlorophenoxy)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]ethan-1-one
3-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)aniline
methyl 6-{[(furan-2-ylmethyl)(methyl)amino]methyl}-3-(2-methylbenzamido)thieno[2,3-b]pyridine-2-carboxylate
{2,2-dimethyl-3-[2-(thiophen-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
ethyl 2-{3-[2-methyl-3-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetate
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
N-[1-(thiophen-2-yl)propyl]-1H-pyrrole-2-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-ethyl-N-(oxolan-2-ylmethyl)butanamide
N-[(2,3-difluorophenyl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
4-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-3-methyl-1H-pyrazole
1-{3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]phenyl}imidazolidin-2-one
2-(3-methyl-3-phenylbutanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrimidin-2-amine
N-{1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
(3S,4R)-4-methyl-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine-3,4-diol
8-(6-aminopyridine-3-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
2-[4-(dimethylamino)phenyl]-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]ethan-1-one
1-cyclopentyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(2-methoxyphenoxy)-1-[3-(methylsulfanyl)butyl]piperidine-4-carboxylic acid
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
2-(2-methoxyphenoxy)-N-{[1-(1,3-thiazol-5-ylmethyl)piperidin-3-yl]methyl}acetamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
(2R,3R,6R)-3-phenyl-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
(1-{3-[(2-amino-5-ethylpyrimidin-4-yl)amino]propyl}piperidin-2-yl)methanol
1-butyl-4-[4-(propan-2-yl)pyrimidin-2-yl]piperazin-2-one
3-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,2-oxazole-3-carboxamide
N-(butan-2-yl)-4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide