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5-chloro-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1,3-dimethyl-1H-pyrazole-4-sulfonamide
N'1-(1-cycloheptylpiperidin-3-yl)cyclopropane-1,1-dicarboxamide
N-(1-benzofuran-2-ylmethyl)-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
1-propyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(piperidine-1-carbonyl)pyridine
5-[(E)-2-phenylethenyl]-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-[(2-fluorophenyl)methyl]-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3,4-dimethylphenyl)methyl]-4-(5-propyl-1,2-oxazole-4-carbonyl)piperazin-2-one
N,8-dimethyl-3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-N,N-dimethylpropane-1-sulfonamide
2-methyl-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenyl)piperazine
2-cyclohexyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-benzoxazole-6-carboxamide
5-(5-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)-1,2-oxazole
3-{2-oxo-4-[3-(thiophen-2-yl)propanoyl]piperazin-1-yl}benzonitrile
4-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)thiomorpholine
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-3-yl)propan-1-one
9-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(1R,5R)-N,N-dimethyl-6-(3-phenyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
9-ethyl-1-methyl-4-{[2-(methylsulfanyl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-6-cyclopropylpyrimidin-4-amine
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2,5-dimethylphenyl)ethan-1-one
3-(4-chloro-2-methylbenzoyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
methyl (2S)-1-(5-benzamido-1-cyclopentyl-1H-1,3-benzodiazole-7-carbonyl)pyrrolidine-2-carboxylate
1-methyl-6-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
(1-benzothiophen-2-ylmethyl)({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
2-[2-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)phenoxy]acetic acid
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(4,4,4-trifluorobutyl)pyrrolidine-2-carboxamide
2-[4-(3-methoxypyrazin-2-yl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
N,N-dimethyl-2-[(1S,5R)-3-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(2-chlorophenyl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]acetamide
N-methyl-N-(1-methylpiperidin-4-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methyl}benzoic acid
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-(1-methyl-1H-pyrazol-4-yl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
11-[benzyl(methyl)amino]-4-[2-(3-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
4-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)phenol
5-(morpholin-4-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-methyl-5-(4-methylpiperidin-1-yl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(benzyloxy)-8-[2-(phenylsulfanyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperazine
4-[4-(2-{[(1-ethylpyrrolidin-2-yl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-{2-methyl-1-[3-(4-methylpyridin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
1-(3-methoxyphenyl)-2,2-dimethyl-4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-6-methylpyridin-2-ol
3-(2,3-dimethoxyphenyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidine