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2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(methylsulfanyl)propyl]acetamide
5-propyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
8-[(2-ethylpyrimidin-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecane
4-[(dimethylamino)methyl]-1-(5-methyl-1,3,4-oxadiazol-2-yl)azepan-4-ol
2-ethoxy-5-{2-[(pyridin-3-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
1-(1-cyclopentanecarbonylpiperidin-3-yl)-4-(2-methylphenyl)piperazine
N-(2-methoxyethyl)-N,5,6-trimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1-(cyclopropylmethyl)-3-(1H-pyrazol-5-yl)piperidine
1-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
methyl 4-({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}carbamoyl)butanoate
4-[(3,5-dimethoxyphenyl)methyl]-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-(2-methoxyethyl)-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(propylsulfanyl)ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(4-methylphenyl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[methyl(1-methylpiperidin-4-yl)amino]ethan-1-one
6-methoxy-4-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(trifluoromethyl)benzamide
N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[5-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
(4aR,7aS)-N,N-dimethyl-4-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
4-amino-2-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidine-5-carbonitrile
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-5-(2-hydroxy-2-methylpropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butane-1,2-dione
1-{2-[1-(2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-1-yl}propan-1-one
2-methoxyethyl 2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxylate
N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
3-benzyl-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
4-(4-methylphenyl)-N-(pyridin-3-ylmethyl)-5-(pyridin-4-yl)pyrimidin-2-amine
4-{3-[(4-methoxyphenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}benzoic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-{6-amino-5-cyano-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridin-2-yl}benzoic acid
(1S,6R)-3-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
4-methyl-2-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-benzoxazole
[5-(1-{1-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-1H-1,2,3-triazol-4-yl)furan-2-yl]methanol
4-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}benzamide
1-{[(2R,5S)-5-(2H-1,3-benzodioxol-5-ylmethyl)oxolan-2-yl]methyl}-4-ethylpiperazine
N-benzyl-N,3-dimethyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-sulfonamide
3-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
N-(2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}ethyl)acetamide
N-[(3S,5S)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
1-ethyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-6-oxopiperidine-3-carboxamide
2-{[2-(benzyloxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane
8-(2-hydroxynaphthalene-1-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[1'-(3-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(morpholin-4-yl)ethan-1-one
1-{4-[(3,5-dichloro-2-methoxyphenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
6-methyl-N4-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]pyrimidine-2,4-diamine