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2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1-benzofuran-7-carboxamide
5-(1H-pyrazol-1-ylmethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}furan-2-carboxamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-[(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)methyl]-1H-indole
N-methyl-2-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyridine-4-carboxamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-phenylethane-1,2-dione
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2-methoxypyrimidin-5-yl)methyl]amine
(2S)-1-(piperidin-4-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}pyrrolidine-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}azepan-2-one
(2S)-3-phenyl-2-({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)propanamide
5-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-(3-fluorophenyl)-2-{4-[2-(4-oxo-1,4-dihydropyridin-1-yl)acetyl]morpholin-3-yl}acetamide
3-methoxy-1-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
3-cyclopropyl-5-[2-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-1,2,4-triazole
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(thiophen-2-ylmethyl)acetamide
(dicyclopropylmethyl)({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(5-methanesulfonamido-2-methylphenyl)-2-(pyridin-3-yl)piperidine-1-carboxamide
(9aS)-N-(3-chloro-2-fluorophenyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
2-ethyl-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
8-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-({1-[4-(3-methylphenyl)phenyl]piperidin-4-yl}amino)butan-1-ol
3-(2-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)pyrrolidin-2-one
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile
methyl (1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
3-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-(3-fluoro-4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N,N-dimethylpropanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(thian-4-yl)piperidine-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(2,3,4-trifluorobenzoyl)piperazin-2-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
4-methoxy-6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
(2S)-2-amino-1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-{3-[(3R,4S)-3-[(2-methylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
1-(4-{[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{2-[(3aS,6aS)-1-(2-ethoxybenzoyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]ethyl}morpholine
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
4-cyclopentyl-3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}piperazin-2-one
2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-amine
2-cyclopentyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)propan-1-one
4-chloro-2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol