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N-[4-methyl-3-(3-methylbenzamido)phenyl]quinoxaline-5-carboxamide
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-N,N-dimethylpiperazine-1-carboxamide
2-[(4-chlorophenyl)methyl]-8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
3-cyclopentyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(3aR,6aR)-2-methanesulfonyl-5-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(butan-2-yl)-N-[(3-methylthiophen-2-yl)methyl]-2-(oxan-4-yl)acetamide
N-(3,4-difluorophenyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-amine
methyl(thiophen-2-ylmethyl){[3-(2-{4-[3-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl}amine
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
{1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3-[(dimethylamino)methyl]piperidin-3-yl}methanol
1'-(4-methoxyphenyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-3-propyl-1H-pyrazole-5-carboxamide
4-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]-4H-1,2,4-triazole
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
1-ethyl-5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amine
4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-phenylpiperazin-2-one
(3aR,6aR)-2-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-chloro-4-{[1-(furan-2-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-cyclopropyl-4-{[1-(1-methyl-1H-pyrazol-4-yl)propyl]sulfamoyl}benzamide
6-methyl-4-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
2-({2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-cyclopropyl-5-(1H-indol-3-ylmethyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-3-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
1,9-dimethyl-4-[(5-methylthiophen-2-yl)sulfonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-benzyl-3-methyl-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)pyridine
2-[1-(2-methylpropyl)-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N-(2-methylpropyl)-3-(1,2-oxazolidin-2-yl)-N-(3-phenylprop-2-yn-1-yl)propanamide
{2H-1,3-benzodioxol-5-yl[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}dimethylamine
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
3-[1-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
5-methanesulfonyl-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-methylpyrimidin-4-amine
(1S,5R)-3-methyl-N-[3-(trifluoromethyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-[2-(4-ethyl-1,4-diazepan-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
(3aS,6aR)-5-cyclobutanecarbonyl-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(1-ethylpiperidin-4-yl)-N-[3-methyl-1-(pyridin-3-yl)butyl]acetamide
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
1-(2,4-dimethoxyphenyl)-4-methylphthalazine
ethyl 1-(3-methylbutyl)-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
4-ethyl-3-({2-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-5-methyl-4H-1,2,4-triazole
N-{[4-(1H-1,3-benzodiazol-6-yl)phenyl]methyl}methanesulfonamide
N-({5-[(2,6-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-phenylquinazoline
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one