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1-(furan-2-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-(1-methanesulfonylpiperidin-4-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
1-{3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propyl}piperidine
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]acetamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
(5S,9aS,9bS)-5-(4-fluoro-3-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(5-fluoro-1H-indol-2-yl)methyl]methylamine
(2R)-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)-3-phenylpropan-1-ol
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
ethyl 4-benzyl-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine-4-carboxylate
3-[3-(1,5-dimethyl-1H-pyrazol-4-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2-[4-(3,5-dimethylbenzoyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
2-[3-(2-methoxyethyl)-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl]benzoic acid
2-hydroxy-5-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
(2R)-2-amino-N,4-dimethyl-N-[(3-methylpyridin-4-yl)methyl]pentanamide
2-(3-fluorophenoxymethyl)-N-methyl-N-(pyrimidin-4-ylmethyl)-1,3-oxazole-4-carboxamide
4-{[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]amino}-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
2-methoxy-5-oxo-6-[2-(oxolan-3-yl)ethyl]-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-[(2-butoxy-3-methoxyphenyl)methyl]pyrrolidin-3-amine
N-[(3R,4S)-4-cyclopropyl-1-[3-(dimethylamino)pyrazin-2-yl]pyrrolidin-3-yl]methanesulfonamide
2-{[4-(3-methylphenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-(dimethylamino)-2-(3-methylphenyl)-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}acetamide
1-(2-methoxyethyl)-3-methyl-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S)-4-methyl-2-{[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazol-3-yl]formamido}pentanamide
N-[(2S)-1-oxo-1-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propan-2-yl]acetamide
4,5-dimethyl-N-(prop-2-en-1-yl)-N-(propan-2-yl)thiophene-2-carboxamide
(1R,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-methylpiperidine
6-(4-chlorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,2-dimethylcyclopropane-1-carboxamide
2-({2-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
N-[(3-fluorophenyl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
propan-2-yl 2-chloro-5-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]acetamido}benzoate
N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-4-carboxamide
(3R,5S)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(3-hydroxyphenyl)acetamide
methyl 1-[2-hydroxy-3-(4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
1-(2H-1,3-benzodioxol-5-yl)-5-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
4-({3-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)thiomorpholine
2-{2-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N,N-bis(propan-2-yl)benzamide
N-[(3S)-2-oxoazepan-3-yl]-4-(4-{[3-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)benzamide
6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide