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N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(pyrrolidin-1-yl)benzamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-methyl-2-oxopyrrolidin-1-yl)acetamide
1-{2-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
(4aS,7aR)-4-acetyl-N-(4-chlorophenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-methyl-1-(3-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propyl)-1H-1,2,3,4-tetrazole
3-({2-[5-(oxan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-5-(propan-2-yl)-1,2,4-oxadiazole
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)-1,4-oxazepane
2-(1,3-benzothiazole-6-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(3-methylcinnolin-5-yl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
4-(4-phenoxybutyl)-1,3λ6,4-oxathiazinane-3,3-dione
2-(4-fluorophenyl)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-ethyl-N-methylacetamide
(1R,5R)-6-[2-(phenylsulfanyl)ethyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
7-propyl-2-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3-methoxypropyl)-1-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidine-3-carboxylic acid
4-[4-ethyl-6-(1H-pyrazol-3-yl)pyrimidin-2-yl]morpholine
5-{[(2-amino-5-methylpyrimidin-4-yl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(2-ethoxy-3-methoxyphenyl)methyl]piperidin-3-amine
9-[(3-chloro-1H-indol-2-yl)methyl]-3-oxa-9-azaspiro[5.5]undecane
1-(2,6-dimethoxypyridin-3-yl)-3-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]urea
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenylpiperidine
1-[2-(dimethylamino)-4-{methyl[3-(1H-pyrazol-1-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5,8-dimethyl-2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}quinolin-4-ol
1-[1-methyl-5-({methyl[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(pyridin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrazole-3-carboxylic acid
5-cyclopropanecarbonyl-1'-[(3-ethenylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)methanol
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-methylacetamide
(3R,4R)-4-cyclobutyl-1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3-methylpiperidin-4-ol
1-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
(2-{1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
4-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)phenol
2-(4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
(2S,4S)-4-amino-N-ethyl-1-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
(4S,4aS,8aS)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-phenyl-decahydroquinolin-4-ol
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
7-(cyclobutylmethyl)-2-(pyridine-3-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-chloro-4-{[4-(dimethylamino)azepan-1-yl]methyl}phenol
N-(1-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}piperidin-4-yl)acetamide
5-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}quinoline
4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}-N-[2-(thiophen-2-yl)ethyl]benzamide
(3aS,6aS)-2-benzyl-5-{2-methylthieno[2,3-d]pyrimidin-4-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,4S)-2-(2-fluorophenyl)-5-[(5-methylthiophen-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-methyl-4-[3-(1H-pyrazol-3-yl)phenyl]aniline