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1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(dimethylamino)methyl]-1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)piperidin-3-ol
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-(dimethylamino)-7-(2-methoxybenzenesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-N-(2,4-dimethylphenyl)-3-oxopropanamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-(2-methylphenoxy)azetidine
ethyl 1-[4-(oxolan-2-ylmethoxy)phenyl]-1H-imidazole-2-carboxylate
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,4-diazepane
3-(3-fluorophenyl)-4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-2-one
4-(2-chlorophenyl)-6-methoxypyrimidin-2-amine
1-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-(2,3-dimethylphenyl)-4-(pyrrolidine-1-carbonyl)pyridine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
1-[6-(cyclopropylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-N,N-diethylpiperidine-4-carboxamide
(2S,4R)-4-amino-1-(2-cyanobenzoyl)-N-methylpyrrolidine-2-carboxamide
7-cyclohexyl-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
(3E)-2-[4-(2-methoxybenzoyl)piperazin-1-yl]hept-3-enoic acid
1-(2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
3-[2-(dimethylamino)ethyl]-8-(2,2-dimethylpropyl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
({4-[(3-chloro-5-fluorophenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
2-{4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
8-(pyrazin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-({[(3,5-dimethyl-1H-indol-2-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
6-methoxy-3-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-methyl-2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenol
(1S,5R)-3-acetyl-N-(4-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(1R,2S)-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-propylcyclopropane-1-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(3-fluoropyridin-2-yl)piperidine-4-carboxylic acid
N-phenyl-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-methoxy-1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]propan-1-one
4-{2-[2-(2,1,3-benzoxadiazol-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
5-methyl-1-(4-methylphenyl)-4-[4-(2-oxopiperidin-1-yl)butanoyl]piperazin-2-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-2-yl}methanol
1,3-dimethyl-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}-1H-pyrazole-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
2-(dimethylamino)-8-[(1-ethyl-1H-indol-4-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-(2-aminoethyl)-5,6-dimethyl-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
4-(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazin-2-one
N-(1H-1,3-benzodiazol-2-yl)-2-{[2-(1H-1,2,4-triazol-1-yl)propyl]amino}acetamide
3-(5-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-{4-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid