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4-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1H-1,2,3-triazole-5-carboxamide
1-(furan-2-ylmethyl)-4-(oxane-2-carbonyl)piperazine
1-propyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazole
4-{[3-(dimethylamino)propyl]amino}-5-methyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]benzene-1,2-diol
1-cyclopentyl-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(4-fluorophenyl)-1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
2-ethoxy-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1,4-diazepane-1-carbaldehyde
7-(cyclopropylmethyl)-N-(2,2-difluoroethyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-ethyl-N-[(3R,4S)-1-[2-(methylcarbamoyl)ethyl]-4-propylpyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
dimethyl({4-methyl-5-[1-(2-propylpyridine-4-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
4-[5-(methanesulfonylmethyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]-2-methylpyridine
5-fluoro-N2-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-N4,N4-dimethylpyrimidine-2,4-diamine
2-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-1,2-oxazinane
2-[5-(6-ethoxypyridin-3-yl)-4-phenyl-1H-imidazol-1-yl]-2-(hydroxymethyl)propane-1,3-diol
1-(furan-2-ylmethyl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)piperidine-4-carboxamide
8-(5-acetylthiophene-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(pyrrolidine-1-carbonyl)pyridine
{2-[4-(2,5-dimethylbenzoyl)morpholin-2-yl]ethyl}dimethylamine
6-(2,3,4-trimethoxyphenyl)-9H-purine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(3,4-difluorophenyl)propanamide
(1R,7S)-N-(furan-2-ylmethyl)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(2-{[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-ethyl-2-[4-(1-ethyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-1-yl]acetamide
5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
N-[2-(4-{2,7-diazaspiro[4.5]decane-7-carbonyl}phenoxy)ethyl]acetamide
N-cyclohexyl-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N-methylbutanamide
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}acetamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-methyl-N-(oxolan-3-yl)-1,3-oxazole-4-carboxamide
7-(2,3-dimethoxyphenyl)-9-methoxy-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-({2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(2-aminoethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[(3,5-difluorophenyl)methyl]-8-(3-fluoropyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-4-(furan-3-yl)-6-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-(1-{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
2-[(3,5-dimethyl-1H-indol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
N-(5-chloro-2-methoxyphenyl)-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
(3S,4S)-4-(pyridin-2-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
{1-[3-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]piperidin-2-yl}methanol
1-{4-[(oxan-2-ylmethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(4aS,8aR)-6-(4-methoxypyrimidin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(2-methyl-5-oxo-1,4-diazepan-1-yl)-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide