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8-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
N-(2-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}ethyl)morpholine-4-carboxamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-(1H-1,3-benzodiazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
N-ethyl-N'-(3-hydroxyphenyl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]butanediamide
[(2-methyl-1H-imidazol-4-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
(3R,4S)-4-(5-methylfuran-2-yl)-1-[1-(piperidin-1-yl)cyclohexanecarbonyl]pyrrolidin-3-amine
1-(4-methoxybenzoyl)-4-(oxane-4-carbonyl)piperazine
2-methyl-N-{1-[1-(2-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[4-(3-methoxyphenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(2-chloro-6-fluorophenyl)-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}acetamide
2-(2-hydroxyethyl)-8-[3-(1-methyl-1H-pyrrol-2-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-(2-methylphenyl)-4-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-yl}piperazine
N-(3-hydroxy-2,2-dimethylpropyl)-2-[(4-methylphenyl)amino]-2-phenylpropanamide
8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-ethyl-2-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[(pyridin-3-ylmethyl)amino]benzamide
ethyl 1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
methyl 1-[(3S,5S)-1-[(2-ethoxyphenyl)methyl]-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2S)-2-amino-1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pentan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
5-tert-butyl-4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)furan-2-carboxamide
3,5-dimethoxy-N-({1-[3-(pyrazin-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
3-[(3R,4S)-3-(4-chloro-1,5-dimethyl-1H-pyrazole-3-amido)-4-cyclopropylpyrrolidin-1-yl]propanoic acid
1,5-dimethyl-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
4-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}piperidin-1-yl)-2-ethylbutan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
5-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
methyl 3-chloro-4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)carbamoyl}amino)benzoate
4-(5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2,4-oxadiazol-3-yl)benzoic acid
(3S,5R)-5-(cyclopropylcarbamoyl)-1-[2-(2-methoxyphenyl)acetyl]piperidine-3-carboxylic acid
5,6-dichloro-2-(oxolan-3-yl)-1H-1,3-benzodiazole
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
(3R,5S)-N-(2-methylpropyl)-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-tert-butyl-2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[2-(trifluoromethyl)morpholine-4-carbonyl]quinoline
1-(1H-imidazol-2-ylmethyl)-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
(3S)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-ol
N-{5-[(2,2-dimethylmorpholin-4-yl)methyl]pyrimidin-2-yl}benzenesulfonamide
N-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-N,2,2,6,6-pentamethylpiperidin-4-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-1,4-dihydroquinolin-4-one
2-[3-(1H-1,2,4-triazol-1-yl)adamantane-1-carbonyl]-2,7-diazaspiro[4.5]decane
N-tert-butyl-3-methyl-2-oxo-N-(pyridin-2-ylmethyl)-2,3-dihydro-1,3-benzoxazole-5-carboxamide