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4-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
1-(4-methanesulfonylphenyl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
2-(furan-3-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-(4-phenyl-1,3-thiazol-2-yl)-2-(trifluoromethyl)morpholine
N,N,4-trimethyl-6-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyrimidin-2-amine
4-[4-(dimethylamino)phenyl]-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]benzamide
1-{1-[2-(benzyloxy)ethyl]piperidin-3-yl}pyrrolidin-2-one
N-[(2-ethoxyphenyl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
1-{1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
{1-[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]piperidin-4-yl}methanol
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
1-[2-(4-methoxyphenyl)ethyl]-5-(4-methoxypiperidine-1-carbonyl)piperidin-2-one
1-[(3-fluorophenyl)methyl]-5-[4-(hydroxymethyl)piperidine-1-carbonyl]piperidin-2-one
[(3R,4S)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4,6-dimethyl-1-(2-oxo-2-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
8-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazol-1-yl}quinoline
3-chloro-N-cyclopropyl-N-({4-[3-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)propoxy]phenyl}methyl)benzamide
{5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
7-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
1-(4-chlorophenyl)-4-{2-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(methylsulfanyl)pyrimidine
N-methyl-4-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3-thiadiazole-5-carboxamide
N-methyl-5-[1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
(1R,5S)-3-(1H-indazole-3-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
[(1-ethylpyrrolidin-2-yl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(1S,5R)-6-(cyclopropylmethyl)-3-[(2,4-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-(morpholin-4-yl)butan-1-one
N-(4-oxo-4H-chromen-6-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
8-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[(2,4-difluorophenyl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
1-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,2-dihydropyridin-2-one
N-cyclobutyl-4-[(furan-3-ylmethyl)sulfamoyl]benzamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(dimethylamino)butanamide
3-[1-(1-methylpiperidin-4-yl)-5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-1H-1,2,4-triazol-3-yl]pyridine
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(furan-2-yl)pyridine-3-carbonitrile
N4-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-(3-oxo-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}propyl)methanesulfonamide
4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
N-({4-hydroxy-1-[2-(3-hydroxyphenyl)acetyl]azepan-4-yl}methyl)benzamide
N-ethyl-5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}pyrimidin-2-amine
[5-(4-phenyl-1-{2-[(pyridin-3-yl)amino]ethyl}-1H-imidazol-5-yl)furan-2-yl]methanol
2-(morpholin-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-3-yl)acetamide
2-{[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]methyl}benzonitrile