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3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyloxan-4-yl)methyl]propanamide
2-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)-8-benzyl-2,8-diazaspiro[5.5]undecane
5-[(2E)-but-2-en-1-yl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
(2E)-3-(furan-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]prop-2-enamide
3-{[(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
(2R,4S)-1-(2,2-diphenylacetyl)-4-hydroxypiperidine-2-carboxylic acid
5-[2-(4-chlorophenoxy)ethyl]pyridin-3-amine
1-[6-(2-methoxyphenoxy)pyridin-3-yl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-5-methylthiophene-2-carboxamide
N-[2-chloro-5-(methylcarbamoyl)phenyl]-4-hydroxy-4-(pyridin-3-yl)piperidine-1-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-3-ethylpiperidine-3-carboxylic acid
N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl)methyl]thiophene-3-carboxamide
4-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethylthiophene-2-carboxamide
2,6-dimethyl-4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}quinoline
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
3-[(7-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
4-{1-[3-(ethylsulfanyl)propanoyl]piperidin-3-yl}benzoic acid
2-amino-1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-methylpropan-1-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
N-ethyl-6-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]pyridine-3-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1-(1,3-benzothiazol-5-yl)-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]urea
methyl 4-{[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylate
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}-N,N-dimethylacetamide
(2S)-2-[2-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-imidazol-1-yl]propanamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
4-[1-(3,4-difluorophenyl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl]pyridine
methyl[(3-methylpyridin-2-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]piperidine-1-sulfonamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-(4-phenyl-1H-imidazol-1-yl)acetamide
2-(2-chloro-6-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-{[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-indole
methyl 5-[(1-methoxy-1-oxopropan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-fluoroethyl)-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
5-chloro-6-(isoquinolin-5-yl)-2-methylpyrimidin-4-ol
methyl[2-methyl-3-(pyrrolidin-1-yl)propyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
2-chloro-3-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-6-methoxyphenol
1-{2-[(E)-2-cyclohexylethenyl]pyrimidin-4-yl}pyrrolidin-3-ol
[(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(2S,4S)-4-amino-N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N,1-dimethylpyrrolidine-2-carboxamide
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
4-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid