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ethyl 1-[(3,5-dimethoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-{4-phenyl-5-[3-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}acetamide
1-[(2-methoxyphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
(2S)-2-cyclohexyl-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]acetic acid
4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
4-{1-[(dimethyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}benzoic acid
(1R,5R)-6-(benzenesulfonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
ethyl 4-(2-methoxyethyl)-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxylate
7-(cyclobutylmethyl)-2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(1H-1,3-benzodiazol-2-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl (2S,4S,5R)-5-(4-chlorophenyl)-1,2-dimethyl-4-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
4-[(5-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
4-(naphthalen-1-ylmethyl)-1,3λ6,4-oxathiazinane-3,3-dione
N-[3-(methylsulfanyl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
3-{1-[2-(2-fluorophenyl)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-(2-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
N-(2-methylpropyl)-1-[(1s,4s)-4-[2-(4-methoxyphenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[3-(2-methylpyrimidin-4-yl)phenyl]pyrrolidine-1-carboxamide
8-{[4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
3-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methoxyphenyl)urea
1-[(2-chloro-6-fluorophenyl)methyl]-1-ethyl-3-(1-ethyl-1H-1,2,3-triazol-4-yl)urea
6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-N,6-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pentan-3-yl)acetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-(2-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-2-yl}ethyl)phenol
N-cyclopropyl-4-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)piperazine-2-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
5-methyl-5-(piperidin-4-yl)-3-(quinolin-8-ylmethyl)imidazolidine-2,4-dione
2-(ethylsulfanyl)-5-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-(3-methoxyphenyl)-N-methylacetamide
8-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-2-methoxyacetamide
2-{1-[(2-chloro-3,6-difluorophenyl)methyl]piperidin-4-yl}-N-methylacetamide
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-N,N-dimethylpyridin-2-amine
3-[4-({[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]carbamoyl}amino)phenyl]-N,N-dimethylpropanamide
6-fluoro-2-[(3-methoxypyrrolidin-1-yl)methyl]quinolin-4-ol
3-(azepane-1-carbonyl)-N-[2-(3-fluorophenyl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2,6-dimethylpyridin-3-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
4-(2-fluorophenoxy)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine-4-carboxylic acid
7-[(2-fluorophenyl)methyl]-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
4-ethyl-3-[1-(3-fluoro-2-methoxybenzoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(3-methylphenyl)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
N-[(1R)-2-hydroxy-1-phenylethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
(3-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}propyl)dimethylamine
2-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
N-(2-methoxyethyl)-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide