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2-(cyclohex-1-en-1-yl)-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
5-[2-(trifluoromethyl)morpholine-4-carbonyl]-3,4-dihydropyrimidin-4-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
5-(1-ethoxyethyl)-1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
5-cyclopropyl-N-methyl-N-(quinolin-5-ylmethyl)-1,2-oxazole-3-carboxamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
2-chloro-5-{1-[2-(3-methylthiophen-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
ethyl 1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
4-{1-[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
5-{[methyl({[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl})amino]methyl}pyrimidin-2-amine
5-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methylpyridine
1-cyclopentyl-N3-methyl-4-oxo-N3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2,2-difluoroethyl)-4-{[2-(1H-pyrrol-1-yl)ethyl]sulfamoyl}benzamide
1,3-dimethyl-5-{3-methyl-1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
3-(4-fluorophenyl)-5-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1H-pyrazole
6-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purin-2-amine
(3R,4S)-4-cyclopropyl-1-(6,8-dimethoxy-4-methylquinolin-2-yl)pyrrolidin-3-amine
3-(3-cyano-4-ethoxyphenyl)-1-ethyl-1-(oxan-4-ylmethyl)urea
7-{4-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]butanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-4-amino-N,N-diethyl-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
3-(3-methoxyphenyl)-5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(2,5-dimethoxyphenyl)-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)acetamide
(1R,5S)-3-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
(4aS,8aS)-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
ethyl 4-[(3-fluorophenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxylate
5-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
N-(2-hydroxyethyl)-N,5-dimethyl-1,3-diphenyl-1H-pyrazole-4-carboxamide
2-{4-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]morpholin-3-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
4-{3,9-diazaspiro[5.6]dodecan-9-yl}pyrimidin-2-amine
1-(adamantan-1-yl)-4-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperazine
2-tert-butyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-ethyl-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}azetidin-3-yl)-1H-1,3-benzodiazole
5-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-(1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}piperidin-3-yl)benzoic acid
dimethyl(3-{2-[1-(quinolin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-(2,5-dimethylphenyl)-3-({5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-yl}formamido)propanamide
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
[(1,3-diphenyl-1H-pyrazol-4-yl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-({4-methyl-5-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
1-[(3-fluorophenyl)methyl]-4-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperazine
2-(methylsulfanyl)-5-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}pyrimidine
5-(3-acetylphenoxymethyl)-N-cyclohexyl-N-(prop-2-yn-1-yl)-1,2-oxazole-3-carboxamide