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2-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1-benzofuran-5-carboxamide
2-(3,5-dichlorophenyl)-5-(4-methylpiperazine-1-carbonyl)pyrimidin-4-ol
6-(2-chlorophenyl)-N-(2,2-difluoroethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(3-{[benzyl(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
N-cyclopropyl-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine-2-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(3-hydroxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
(5-{[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}furan-2-yl)methanol
3-[3-({[1-(4-chlorophenyl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
2-methyl-1-[5-(trifluoromethyl)pyridin-2-yl]-1,4-diazepan-5-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}thian-4-amine
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-propyl-1,3-thiazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(4-ethoxyphenyl)propanamido]acetic acid
N-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)thiomorpholine-4-carboxamide
({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]isoquinoline
2-[4-(2-aminophenyl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
3-ethyl-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylic acid
2-{1-[1-(6-chloroquinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-butyl-1-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazin-2-one
1-(2-methoxyphenyl)-2,2-dimethyl-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazine
1-(2,3-dihydro-1H-inden-2-yl)-5-[(5-methyl-1H-pyrazol-1-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
(4aR,7aS)-N,N-diethyl-6,6-dioxo-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(4aR,7aS)-1-ethyl-4-{[5-(2-fluorophenyl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-chlorophenyl)methyl]-3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)propanamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}benzamide
6-(2-chlorophenyl)-2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2,5-dimethyl-N-[3-(propan-2-yloxy)propyl]-1,3-thiazole-4-carboxamide
(1R,5S,8R)-N-[2,5-difluoro-4-(trifluoromethyl)phenyl]-8-(dimethylamino)-3-azabicyclo[3.2.1]octane-3-carboxamide
N-[(3S,4R)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
5-{1H-pyrrolo[3,2-c]pyridin-4-yl}-1,2,3,4-tetrahydroisoquinoline
5-(dimethylamino)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,3-dihydropyridazin-3-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-(3-hydroxyazetidin-1-yl)ethan-1-one
2-{4-[3-(1-ethyl-1H-pyrazol-3-yl)phenyl]phenyl}-N,N-dimethylacetamide
3-methoxy-1-[7-(1,2,3,4-tetrahydroquinoline-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
4-[(2,2-difluoroethyl)sulfamoyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-ethyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}piperidine-2-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
pyridin-2-yl[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]methanol
2-{2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-(3-methoxyphenyl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
1,5-dimethyl-4-{[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-1,8-naphthyridine-2-carboxamide
4-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
N-cyclopropyl-2-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide