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4-{2-[(6-methyl-2-phenylpyrimidin-4-yl)oxy]hex-5-en-1-yl}morpholine
3-(morpholine-4-carbonyl)-N-[2-(1,3-thiazol-4-yl)ethyl]benzene-1-sulfonamide
4-(2-methoxyethyl)-1-(2-phenylquinazolin-4-yl)piperidine-4-carboxylic acid
4-({2-[1-(2-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[3-(1H-indol-1-yl)propyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(4aR,8aR)-4-[3-(pyrrolidine-1-carbonyl)benzenesulfonyl]-octahydro-2H-1,4-benzoxazine
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-[2-(oxan-4-yl)ethyl]propanamide
2-ethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}benzamide
4-cyclopentyl-3-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-[2-(benzylsulfanyl)ethyl]oxolane-3-carboxamide
2,5-dioxo-6-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
[(3R,4R)-1-(1,3-benzothiazol-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-[(4aR,7aS)-6,6-dioxo-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(2S,4S)-4-[(adamantan-2-yl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
(3S,4S)-4-methyl-1-(4-phenoxybutyl)piperidine-3,4-diol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3S,4S)-4-ethoxypyrrolidin-3-yl]acetamide
N-cyclopropyl-3-methyl-N-[(5-methylthiophen-2-yl)methyl]but-2-enamide
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
2-(2H-1,3-benzodioxol-5-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{3-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}methanesulfonamide
5-[({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2,2,2-trifluoroethyl)acetamide
N-methyl-1-(oxolan-2-ylmethyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(morpholin-4-yl)benzamide
N-(4-{[(1-hydroxybutan-2-yl)(thiophen-2-ylmethyl)amino]methyl}phenyl)acetamide
8-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
1-cyclopropanecarbonyl-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
6-(3-chlorophenyl)-N-(2-methoxyethyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
4-methoxy-6-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-3-methoxyphenol
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}propanamide
1-(2-ethoxyethyl)-N-[(2-methylphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(methoxymethyl)-5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
2-[4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}thiophene-2-sulfonamide
N-(1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
1-(2-{[(5-ethyl-2,6-dimethylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
(2S,4R)-N-cyclopropyl-1-(2,2-diphenylethyl)-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
4-{2-methyl-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]propan-2-yl}morpholine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-[(2,4,6-trimethylphenyl)methyl]pyrrolidine-2-carboxamide
3-[5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazol-1-yl]propanamide
3-{4-[1-(3-phenylpropyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}-1λ6-thiolane-1,1-dione
9-(2,5-dihydro-1H-pyrrole-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2-fluorophenyl)ethyl]-6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carboxamide