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2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methylacetamide
3-(1H-imidazol-1-ylmethyl)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
2-[(2E)-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
1-(2-{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
N,N-dimethyl-2-[4-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperazin-1-yl]acetamide
propyl 4-{[2-(3-methoxyphenyl)phenyl]carbamoyl}piperidine-1-carboxylate
5-(2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-6,8-dimethylquinolin-4-ol
2-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
1-(6-hydroxy-4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)propan-1-one
(4aS,7aR)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-1H-indole
({5-[2-(benzyloxy)phenyl]-1,2,4-oxadiazol-3-yl}methyl)dimethylamine
5-oxo-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}pyrrolidine-3-carboxylic acid
N-[(5-chlorothiophen-2-yl)methyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
N,N,4-trimethyl-5-[4-(1H-1,2,4-triazole-3-carbonyl)piperazine-1-carbonyl]pyrimidin-2-amine
5-hydroxy-6-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
4-(1-{2-[5-(2-methylpropyl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)pyrimidine
5-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
(3R,5R)-N-(oxolan-2-ylmethyl)-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
5-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N'-[(1-cyclopentylpyrrolidin-3-yl)methyl]-N,N-diethylethanediamide
4-[2-(2,2-diphenylethyl)morpholin-4-yl]butan-1-ol
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(quinolin-4-yl)pyrrolidin-3-yl]sulfamoyl})amine
2-(ethylamino)-N-[1-(phenylcarbamoyl)piperidin-4-yl]pyrimidine-5-carboxamide
2-[4-(2-methoxyphenoxy)piperidin-1-yl]pyrimidin-4-amine
1-benzoyl-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(1R,3S)-3-(2,3-dihydro-1H-isoindole-2-carbonyl)-N,N,2,2,3-pentamethylcyclopentane-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-4-(pyridin-4-yl)pyrimidin-2-amine
1-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
3-({[(dimethyl-1,2-oxazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
8-{[2-(difluoromethoxy)phenyl]methyl}-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
N-[4-(2-fluorophenoxy)phenyl]-1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
9-[4-(dimethylamino)benzoyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)acetamide
1-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-3-phenylpropan-1-ol
3-(3-methoxyquinoxalin-2-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
N2-benzyl-6-[2-(methylsulfanyl)phenyl]-1,3,5-triazine-2,4-diamine
1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-(9H-fluoren-9-yl)-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-4-methyl-1H-1,3-benzodiazole
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-phenoxyfuran-2-carboxamide
3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
9-(2-methoxyethyl)-1-methyl-4-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1,4,9-triazaspiro[5.6]dodecan-10-one