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2-cyclopropyl-9-(oxan-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
methyl 5-cyano-6-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-methylpyridine-3-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-8-[3-(methylsulfanyl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-methoxy-4-(pyridin-3-yl)phenyl]acetamide
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-({2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)pyridine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
methyl (2S)-1-[2-(4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
2-ethyl-5-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
N-butyl-2-ethyl-N-(furan-2-ylmethyl)pyrimidine-5-carboxamide
1-ethyl-N-[2-(3-methoxyphenyl)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[3-(difluoromethoxy)phenyl]methyl}azepan-2-one
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
4-{5-methyl-2-oxo-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}benzonitrile
(2S,4S)-N,1-diethyl-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-amido]pyrrolidine-2-carboxamide
4-(2-methoxyphenoxy)-1-(2-methyloxolane-2-carbonyl)piperidine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl})amine
N-(adamantan-1-yl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
4-(2,6-dimethylpyridin-3-yl)-N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)pyrimidin-2-amine
2-[3-(2-methoxyethyl)-5-[2-(pyridin-4-yl)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl]acetic acid
3-[5-(4-chlorobenzenesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
4-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}piperidine
2-methoxy-5-[(3-propoxypiperidin-1-yl)methyl]benzoic acid
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
(1R,5R)-6-[2-(benzyloxy)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{3-[ethyl(methyl)amino]butyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[4-(3-methoxyphenyl)piperazin-1-yl]-2-(pyrrolidin-3-yl)ethan-1-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(1H-indol-3-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]propanamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(phenylsulfanyl)acetamide
N,N-dimethyl-1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]azepan-4-amine
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-chloro-6-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]pyridine-3-carboxylic acid
[(5-chlorothiophen-2-yl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(1R,5R)-6-(cyclobutylmethyl)-3-(5-propyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
9-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-[(2,4-dichlorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
1-(furan-2-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]piperidine-4-carboxamide
8-(3-chloro-4-ethoxyphenyl)-2-(dimethylamino)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
2-(4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazin-1-yl)pyrimidine
5-[(2-phenylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-(4-fluorophenyl)-N-(1H-indol-2-ylmethyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-[(dimethylamino)methyl]-1-[2-(4-methylphenoxymethyl)furan-3-carbonyl]pyrrolidin-3-ol
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
4-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholine
1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine
(2R,4S)-4-hydroxy-1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidine-2-carboxylic acid