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3-(3-methoxyphenoxy)-1-(4-propylbenzoyl)azetidine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
5,6-dimethyl-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1,2-dihydropyridin-2-one
2-(5-chloro-2-ethoxyphenyl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
1-[2-benzyl-4-(4-methylphenyl)-5-oxopiperazin-1-yl]pentane-1,2-dione
1-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)butan-2-ol
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-methylpyrimidine-5-carboxamide
(4aS,8aR)-6-(1-ethyl-1H-pyrazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
[(1,4-dimethyl-1H-pyrazol-5-yl)methyl][(8-methoxyquinolin-5-yl)methyl]methylamine
(1R,2S,4R)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-(2-phenylethyl)-4-(thiophen-2-ylmethyl)morpholine
2-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-N-(propan-2-yl)pyridine-4-carboxamide
2-{2-[(3R)-3-methylpiperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
2,4-dimethyl-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1,3-oxazole-5-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(4-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenyl)acetamide
5-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[5-(1-carboxy-1-methylethyl)-4-(morpholin-4-yl)pyrimidin-2-yl]piperidine-3-carboxylic acid
(2S)-2-acetamido-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(methylsulfanyl)butanamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
2-{[4-methyl-1-(5-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
ethyl({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
7-(3-chlorophenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-methyl-13-(5-methyl-1-propyl-1H-pyrazol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-cyclohexanecarbonyl-N-ethyl-N-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
1-(propan-2-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
2-(1-phenylmethanesulfonylpyrrolidin-2-yl)pyridine
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-N'-(4-fluorophenyl)ethanediamide
3-(4-ethyl-1H-pyrazol-5-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidine
5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-N-ethylpyrimidin-2-amine
3-{5-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(furan-2-ylmethyl)acetamide
(2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-4-yl)methanol
3-{[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]methyl}benzonitrile
N'-cycloheptyl-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]butanediamide
N-[(4-fluorophenyl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)azepane-2-carboxamide
N-benzyl-N-(cyclopropylmethyl)-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
methyl 5-[4-(1,3-oxazol-5-yl)benzenesulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2,6,8-trimethyl-4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]quinoline
(1R,3s,6r,8S)-4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-azatricyclo[4.3.1.13,8]undecane
2,2,6,6-tetramethyl-N-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-amine
N-{2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}acetamide
[4-({4-[methyl(phenyl)amino]phenyl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl](pyridin-3-yl)methanol
2-(methylamino)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1,3-thiazole-4-carboxamide
2-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-4-(propan-2-yl)-1,3-thiazole
2-[2-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)phenoxy]acetic acid