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(3S,4R)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
6-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile
2-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)benzonitrile
2-(piperidin-1-yl)-N-[2-(pyrazin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
7-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-methyl-6-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-methyl-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(2S,4S)-N-cyclopropyl-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
2-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
7-hydroxy-6-methoxy-4-{2-phenylimidazo[1,2-a]pyridin-3-yl}-1,2,3,4-tetrahydroquinolin-2-one
N-[1-(pyridin-3-yl)propan-2-yl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-{2-methoxy-5-[(4-methylpiperidin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}acetamide
3-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]urea
4-{[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
N-[3-(4-fluorophenyl)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-1,3-thiazol-4-yl}methanol
N,N-dimethyl-1-[(5-propylfuran-2-yl)methyl]piperidin-3-amine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
5-(2-methoxyphenoxymethyl)-N-(1,2-oxazol-5-ylmethyl)-1H-pyrazole-3-carboxamide
4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(piperidin-3-yl)benzamide
4-[(diethylamino)methyl]-5-ethyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)propanamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]propanamide
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
(1R,5S,8S)-N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-8-methoxy-3-azabicyclo[3.2.1]octane-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
3-{5-[(2R)-2-amino-3-phenylpropanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopropylpropanamide
3-chloro-N-[1-(cyclohex-1-en-1-yl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-4-methylpiperazine
[1-({1-[2-(difluoromethoxy)benzoyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N,N-diethyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
(4aS,8aR)-6-(1H-1,3-benzodiazole-5-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
3-(6,7-dimethoxy-4-methylquinolin-2-yl)propan-1-ol
4-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidine-4-carbonyl}morpholine
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methylbenzamide
1-methyl-6-(propan-2-yl)-3-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]-1,2-dihydropyridin-2-one
2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1H-imidazole
3-{[1-(pyrazin-2-yl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
(2S)-2-[3-(azocan-1-yl)propanamido]-2-cyclopropylacetic acid
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(1-methyl-6-oxo-1,6-dihydropyridazin-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-[(2S)-1-acetylpyrrolidine-2-carbonyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylic acid
1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
2-(4-fluorophenoxymethyl)-N-methyl-N-(3-methylbutyl)-1,3-oxazole-4-carboxamide
3-(3-methoxyphenoxymethyl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine