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8-[(3-acetyl-2,4,6-trimethylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]benzamide
3-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-3-yl)propanamide
7-{furo[3,2-c]pyridin-4-yl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-ethoxypyridazine
N-(6-chloropyridin-3-yl)-2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
1-(pyridin-4-yl)-4-[(2R)-pyrrolidine-2-carbonyl]piperazine
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N,2,6,8-tetramethylquinoline-4-carboxamide
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
(2R,3R,6R)-5-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(1R,2R,6S,7S)-4-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pent-4-enamide
4-ethyl-3-{2-[2-(2-fluoro-4,5-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
3-{2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methylimidazolidine-2,4-dione
1-methyl-3-(2-methylpropyl)-N-[1-(4-methylpyridin-2-yl)propyl]-1H-pyrazole-5-carboxamide
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-{4-[(oxolan-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-[2-(azepan-1-yl)ethyl]-3-acetamido-N-(propan-2-yl)propanamide
6-oxo-4-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
1-[(5-{1-[2-(ethylsulfanyl)ethyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl})amine
6-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-3-yl}pyrimidin-4-ol
2-fluoro-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
5-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-(4-fluorophenyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
3-{[butyl(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(3aS,6aS)-2-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{3-[4-(2-methoxyethyl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-(2-chloro-4-fluorophenoxymethyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(1S,5R)-3-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3R,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-{2-methyl-6-[4-(3-methylpyridin-4-yl)piperazin-1-yl]pyrimidin-4-yl}ethan-1-amine
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(furan-3-yl)-1H-imidazole
(1R,5R)-6-benzyl-3-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-fluoro-N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-methylquinoline-4-carboxamide
4-ethyl-1-methyl-3-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]pyrimidine-5-carboxamide
2-methoxy-N-({5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N-cyclopentylpropanamide
2-{2-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-[(2R,3R)-2-hydroxy-1'-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide