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N-[(3-chloro-4-fluorophenyl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
2-(dimethylamino)-N-(1-methanesulfonylpiperidin-4-yl)-2-(3-methylphenyl)acetamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}benzamide
(3E)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]hex-3-enamide
N-{[(3S,4S)-3-hydroxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl]methyl}-2,2-dimethylpropanamide
2-cyclopropyl-4-methyl-N-(1,2-oxazol-3-ylmethyl)pyrimidine-5-carboxamide
2-(2,4-difluorophenyl)-5-(4-fluorobenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[(1-hydroxycyclohexyl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
7-[2-(2-methoxyethoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-5-ethyl-2-methylpyrimidin-4-amine
(3S,7S,8aS)-7-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-fluoro-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
(2S,4S)-4-amino-N-ethyl-1-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidine-2-carboxamide
(1R,5R)-3-(5-chlorothiophene-2-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
1-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
5-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-N,N-dimethylpyridin-2-amine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(2-ethyl-1H-1,3-benzodiazol-1-yl)propan-1-one
(3R,5S)-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-3-ol
N-(2-hydroxyethyl)-3-methyl-N-[(3-methylthiophen-2-yl)methyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]oxane-4-carboxamide
1-(2-hydroxyethyl)-N-propyl-N-(pyridin-3-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-(2-chlorophenyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-phenylpropanamide
8-(1H-indol-2-ylmethyl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(piperidine-1-carbonyl)pyridine
N-{2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}acetamide
(2S)-2-amino-N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-3-(1,3-thiazol-4-yl)propanamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-hydroxyphenyl)ethan-1-one
9-methyl-3-(1-propyl-1H-pyrazole-5-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
4-[5-({2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
N-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
N-cyclohexyl-3-[2-(furan-2-yl)-2-oxoacetamido]-2-methylbenzamide
N-(furan-2-ylmethyl)-2-(4-methanesulfonylphenyl)-N-(3-methylbutan-2-yl)acetamide
(2S)-N-ethyl-1-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)pyrrolidine-2-carboxamide
(1R,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3-methoxypropyl)-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(4-methylphenoxy)piperidine
methyl 1-[2-hydroxy-3-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
3-[({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-N,N-dimethylbenzamide
N-[3-(3-fluorophenyl)phenyl]-1-(1,3-oxazole-5-carbonyl)piperidine-4-carboxamide
3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
1-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-2-methylpropan-1-ol
{3-[(5-ethylfuran-2-yl)methyl]-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-{[(1-carbamoylethyl)(methyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-cyclobutyl-1-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one