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(3S,4S)-3-hydroxy-4-(propan-2-yloxy)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-1-carboxamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-[(2-aminopyridin-3-yl)methyl]-8-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2-methoxyethyl)-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
1-(4-fluorophenyl)-4-(morpholine-2-carbonyl)-1,4-diazepane
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
N-cyclopropyl-1-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3R,4R)-3-[ethyl(3-methylbut-2-en-1-yl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2H-1,3-benzodioxole-5-carboxamide
N-{[(2S,4S)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide
4-[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2,6-dimethoxypyrimidine
N,N-diethyl-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carboxamide
4-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)thiomorpholine
2-({2-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2-methoxyethoxy)ethan-1-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(4-methylquinolin-2-yl)piperidin-3-ol
1-(2-methoxypyridine-4-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-chloro-2-oxo-1,2-dihydropyridine-3-carboxamide
6-{[methyl(prop-2-en-1-yl)amino]methyl}-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-5-yl)-3-{[(2-methyl-1H-imidazol-4-yl)methyl]amino}-5-(methylsulfamoyl)benzamide
3-[1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazol-3-yl)-N-methylformamido]-N-methylpropanamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
[(5-chloro-2-methoxyphenyl)methyl](ethyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
N-[2-(azepane-1-carbonyl)phenyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
2-({[(1-ethyl-1H-indol-6-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
9-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-6-oxa-9-azaspiro[4.5]decane
1-[2-(1H-imidazol-4-yl)ethyl]-2-(1-phenylethyl)-1H-imidazole
(3S,4S)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3,4-diol
4-{[5-(2-amino-6-methylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}piperazin-2-one
2-(dimethyl-1,3-thiazol-5-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-benzyl-3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidine-1-carboxamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-ethyl-5-(2-ethylpiperidine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
(1R,3S)-7-[(3-methylphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
2-{2-[(4-phenylazepan-1-yl)methyl]phenoxy}acetic acid
(1S,5R)-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-chloro-4-[({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-6-methoxyphenol
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-[4-(morpholin-4-yl)butyl]acetamide
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)propanamide
N-[(5-chloro-2-propoxyphenyl)methyl]-9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-3-(N-methylmethanesulfonamido)propanamide
8-(3-hydroxypropyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-oxo-2-(propan-2-yl)-1,6-dihydropyrimidine-5-carboxamide
1-(2-methoxyphenyl)-4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}piperazine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-methylpiperidin-2-one