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3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-methylpyridine-3-carbonitrile
N-[3-chloro-2-(propan-2-yloxy)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
3-(2-methoxyethyl)-5-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-(1,2-oxazol-3-ylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N,N-dimethyl-5-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)furan-2-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
5-cyclopropyl-N-(1-methoxybutan-2-yl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(1H-1,2,4-triazol-5-yl)ethyl]amine
N-[(2-amino-1,3-thiazol-4-yl)methyl]-N'-[2-(propan-2-yl)phenyl]butanediamide
2-(propan-2-yl)-1-[(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazol-5-yl)methyl]-1H-imidazole
N-(2,5-difluorophenyl)-2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-({[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]formamido}methyl)-N-methylfuran-2-carboxamide
(3S,4S)-4-(propan-2-yl)-1-(4-sulfamoylbutanoyl)pyrrolidine-3-carboxylic acid
(3S,4R)-4-(hydroxymethyl)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-ol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)but-3-enamide
3-[1-(2-oxo-1,2-dihydroquinolin-4-yl)-N-(pyridin-3-ylmethyl)formamido]propanoic acid
1-(2-methoxyethyl)-3-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{5-[3-(methylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)-1H-pyrazole
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1-(propan-2-yl)-1H-pyrazole-3-carboxamide
2,6-dimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
4-[5-(methoxymethyl)-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
4-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-[1-(4-chlorophenyl)ethyl]-1,3-oxazole-4-carboxamide
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine
4-(4-phenyl-1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
4-chloro-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-[2-(pyridin-4-yl)phenyl]cyclopropanecarboxamide
6-methoxy-N,3-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxylic acid
1-[1-(4-fluorophenyl)propan-2-yl]-4-methyl-1,4-diazepan-5-one
N-[(2R,4S,6S)-2-(3-hydroxyphenyl)-6-(1-methyl-1H-1,2,3-benzotriazol-5-yl)oxan-4-yl]acetamide
7-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-3,4-dihydro-2H-1-benzopyran-4-one
3-fluoro-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyridin-4-amine
2-methyl-6-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,3-dihydropyridazin-3-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2,2,2-trifluoroethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-(3-methanesulfonamido-4-methoxyphenyl)-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
(4aS,8aR)-1-(2-aminoethyl)-6-(1-benzofuran-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[(4-methoxypiperidin-1-yl)methyl]-6-methylquinolin-4-ol
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-[(2-methoxy-3,5-dimethylphenyl)methyl]-1-(methoxymethyl)-N-methylcyclopropan-1-amine
N-cyclohexyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
2-methyl-3-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole