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(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aS,8aR)-1-[2-(ethylsulfanyl)ethyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-oxo-4H-chromene-2-carboxamide
(3S,4R)-1-[3-(2-ethoxyethoxy)benzoyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
6-amino-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
(3S)-3-{[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}azepan-2-one
4-hydroxy-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
5-{4-[2-(3-methoxyphenoxy)ethyl]piperazine-1-carbonyl}-2,4-dimethylpyrimidine
4-[(1-{[1-(thian-4-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazol-2-amine
8-(1H-indol-3-ylmethyl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-chlorophenoxy)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
3-methyl-1-(2-methylpropyl)-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1,2-dihydroquinoxalin-2-one
(3S,4R)-3-benzyl-4-methyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-ol
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
(1S,5R)-6-(1H-imidazol-2-ylmethyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
N-[5-(2-methoxyacetamido)-2-methylphenyl]-3-(3-methylphenoxy)azetidine-1-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-methyl-7-(2-phenylquinolin-4-yl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-3-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-methoxyfuran-2-carboxamide
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]cyclopropanecarboxamide
5-methoxy-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-indole-2-carboxamide
3-{[1-(2-hydroxyphenyl)ethyl]carbamoyl}benzoic acid
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-{1-[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
(3R,5R)-N-butyl-1-[(3,4-dimethoxyphenyl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(azepane-1-carbonyl)-N-cyclopentyl-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(difluoromethoxy)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-5-phenylpentan-1-one
1-(cyclopropylmethyl)-3-[(3,4-dimethoxypyridin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-5-propyl-1,2-oxazole-3-carboxamide
1-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)-3-(pyrrolidine-1-carbonyl)piperidine
N-(3-methoxypropyl)-1-methyl-N-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-amine
N-(3-chloro-4-propanamidophenyl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-benzyl-1-cyclohexyl-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-3,4-dihydroxy-N-(2-phenylphenyl)piperidine-1-carboxamide
1-[(3-methylphenyl)methyl]-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)acetamide
[(3aS,6aS)-2-(2-propyl-1,3-thiazole-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol