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2-(4-fluorophenyl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]benzamide
4-cyclobutyl-6-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
5-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[2-(3,4-difluorophenyl)ethyl]-1-(propane-2-sulfonyl)piperidine
dimethyl[1-(4-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}phenyl)ethyl]amine
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[4-(2,3-dimethoxy-5-methylphenyl)phenyl]methyl}piperidine
3-[5-(5-fluoro-2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
2-(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
2-ethyl-4-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,3-oxazole-5-carboxamide
3-(cyclopropylmethyl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine-3-carboxylic acid
4-(1-methyl-1H-imidazol-2-yl)-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(6-methylpyridin-2-yl)methyl]acetamide
4-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)piperidin-2-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-methyl-6-[(4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-ol
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
2-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,2-oxazinane
(3aR,6aR)-2-cyclopentyl-5-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-pyrazol-5-yl)acetamide
4-methanesulfonyl-N-(2-methyl-2H-1,2,3-benzotriazol-4-yl)piperazine-1-carboxamide
methyl 4-({2-[2-(cyclopropylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1H-pyrazole-3-carboxylate
(3R,4R)-4-ethyl-1-[4-(methylsulfanyl)benzoyl]piperidine-3,4-diol
N-(6-cyanopyridin-3-yl)-4-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
5-[(9-ethyl-9H-carbazol-3-yl)methyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyridine-3-carboxamide
4-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]thiophene-2-carboxamide
N3-cyclopentyl-1-(3-methylbutyl)-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-4-(trifluoromethyl)benzamide
7-[(2,3-difluorophenyl)methyl]-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
4-(2-methoxyphenyl)-2-methyl-1-(5-phenyl-1,3-oxazole-4-carbonyl)piperazine
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-3-cyclopropylpropanamide
methyl 2-(2-aminopyrimidin-5-yl)benzoate
4-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
methyl 4-[4-(4,4,4-trifluorobutanoyl)piperazin-1-yl]benzoate
1-[2-(methylsulfanyl)benzoyl]piperidine-4-carbonitrile
3-methyl-5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
6-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
9-(2-fluoro-4-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1,4-diazepane-1-sulfonyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
5-[benzyl(methyl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
2-(2,3-dihydroxypropyl)-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
1'-(2,3-dihydro-1-benzofuran-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]