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N-{4-fluoro-3-[({[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}carbamoyl)amino]phenyl}acetamide
1-(propan-2-yl)-4-(1,3-thiazole-4-carbonyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
5-[3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
2-{5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-ol
2-ethyl-N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]butanamide
1-({[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}methyl)cyclopentane-1-carboxylic acid
5-{3-[4-(3-hydroxyphenyl)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
2,4,5-trimethoxy-N-[(1-methylpiperidin-3-yl)methyl]benzamide
2-methoxy-6-{[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
N-methyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(oxan-2-ylmethyl)butanamide
4-(5-acetylthiophene-3-carbonyl)-6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
(3S,4R)-3-ethyl-1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-methylpiperidin-4-ol
2-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-6-methoxyphenol
1-[(3-fluorophenyl)methyl]-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]-6-oxopiperidine-3-carboxamide
4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-propyl-1,3-thiazole
5-(2-fluorophenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(1,3-benzothiazol-2-yl)-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}pyrrolidine-1-carboxamide
2-amino-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(trifluoromethyl)pyrimidine-5-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
6-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methylpiperazin-1-yl)propan-1-one
2-{3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
1-(5-chloropyrimidin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(2-chloro-6-fluorophenyl)methyl]-5-(methoxymethyl)furan-2-carboxamide
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(2S,4S)-N-ethyl-1-(2-propoxyethyl)-4-[4-(1H-pyrazol-4-yl)butanamido]pyrrolidine-2-carboxamide
8-(1-ethyl-1H-1,2,4-triazol-5-yl)-2-(morpholin-4-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-(oxolan-2-ylmethyl)-5,5-diphenylpiperidin-2-one
6-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
8-(4-aminopyrimidin-2-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
4-(cyclopropylmethyl)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
4-[1-(3-methylpyrazin-2-yl)piperidine-3-carbonyl]morpholine
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]acetamide
5-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]-1-cyclopentyl-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(3R,4R)-4-amino-1-(3-methoxy-2-methylbenzoyl)piperidin-3-ol
N-[(3R,4R)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-(3-hydroxypropyl)-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine-3-carboxamide
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
N-[(3,5-difluorophenyl)methyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
6-chloro-N-{2-[(pyridin-3-yl)amino]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
(2S,4S)-4-amino-1-(3,5-dihydroxy-4-methylbenzoyl)-N,N-diethylpyrrolidine-2-carboxamide