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5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
6-ethyl-2-(morpholin-4-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrimidin-4-amine
2-[ethyl(methyl)amino]-1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]ethan-1-one
(1R,5S)-6-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}-6-azabicyclo[3.2.1]octane
5-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}pyrimidin-2-amine
4-[3-(1-methoxyethyl)phenyl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
(3R,4R)-4-cyclopropyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methylpiperidin-4-ol
1-methyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole-6-carboxamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-chlorophenyl)ethan-1-one
N-[2-(2-chlorophenyl)-1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
1-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-1-carbonyl)cyclopropan-1-amine
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}urea
N-(2-{5-[(2,3-dihydroxypropyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(4-methylphenyl)propanamide
1-ethyl-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
(4aR,7aS)-1-(3-methylbutanoyl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
N-{3-[(cyclooctylamino)methyl]-5-(pyrrolidine-1-carbonyl)phenyl}pyridine-2-carboxamide
2-(dimethylamino)-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-benzyl-2-(4-{4-[methyl(quinolin-5-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}-3-(pyrrolidine-1-carbonyl)pyridine
3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridazine
2,4,5-trimethyl-6-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]pyrimidine
2-cyclopropyl-9-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)thiophen-2-yl]ethan-1-one
1-(2-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-methoxyethyl)amino]methyl}piperidin-2-one
4-(6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyrimidin-4-yl)morpholine
4-[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-1-phenylbutan-1-one
5-butyl-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-methylpiperidine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(2-methyl-1H-imidazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-benzyl-1-methyl-5-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(4-methanesulfonylphenyl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(3S,4S)-4-ethoxypyrrolidin-3-yl]-5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(3-methoxypropyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
8-(dimethyl-1,3-thiazole-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
8-{[3-(trifluoromethyl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(3S,4S)-1-[(3,5-dichloro-4-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
(4aS,7aR)-1-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-1-methylpiperidine-4-carboxamide
5-[(R)-methoxy(phenyl)methyl]-1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazole
2-[(1,3-benzothiazol-2-yl)amino]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N3-methyl-N5-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]pyrrolidin-3-ol
2-methoxy-N-[7-methoxy-2-oxo-4-(quinolin-4-yl)-1,2,3,4-tetrahydroquinolin-6-yl]acetamide
1-(oxolane-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
2-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-(1H-pyrrol-1-yl)propanamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-(azepan-1-yl)-3-[4-chloro-2-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol