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2-amino-N-(2,3-dihydro-1H-inden-2-yl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{4-[(5-butylthiophen-2-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylacetamide
1-ethyl-8-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[3-(1H-imidazol-1-yl)propyl]urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2-ethylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N,N-diethyl-7-[(2-ethylpyrimidin-4-yl)methyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[2-(benzylsulfanyl)ethyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
6-methoxy-N,3-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-benzofuran-2-carboxamide
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-[(3-ethyl-3-hydroxypiperidin-1-yl)methyl]benzoic acid
ethyl 4-[7-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-5-carbonyl]piperazine-1-carboxylate
5-[4-(1,3-benzothiazole-5-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
7-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(2,4-dihydroxyphenyl)methyl]-2-(1-methylpiperidin-2-yl)acetamide
1,7-dimethyl-2-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1H-indole
2-methyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,4-dihydroquinolin-4-one
2-fluoro-N-(isoquinolin-5-ylmethyl)-N-methyl-5-sulfamoylbenzamide
N-methyl-N-(2-methylpropyl)-6-(piperidin-3-yl)pyrimidin-4-amine
(4-benzyl-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-2-yl)methanol
3-(2-amino-1,3-thiazol-4-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
2-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-(3-methoxyphenyl)-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-4-yl]propanamide
1-{4-[(2-phenylethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
ethyl 2-{4-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]piperazin-1-yl}acetate
2-[(6-ethoxyquinolin-2-yl)methyl]-9-oxa-2-azaspiro[5.5]undecane
N-(2-chloro-6-methylphenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
4-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(methylamino)acetamide
methyl 5-[(butan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-(pyrazin-2-yl)-6-[2-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
3-cyclopropyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-(cyclohexylmethyl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]morpholin-3-yl}acetic acid
N-butyl-4-(morpholin-4-yl)pyridine-2-carboxamide
4-({2-[4-(piperidin-1-yl)butoxy]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
(1R,5R)-6-(2H-1,3-benzodioxol-5-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3aR,6aR)-2-methanesulfonyl-5-(4-phenoxybutyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-fluoro-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)naphthalen-2-ol
N-[(3S,4R)-1-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-(2-methyl-1-benzofuran-5-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]urea
7-[(2,3-dimethoxyphenyl)methyl]-2-(furan-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[5-({1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
4-[(2,3-difluorophenyl)methyl]-3-{2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-{4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}ethan-1-one
7-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-methyl-2-(5-methyl-1H-pyrazol-1-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-(2-{4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazin-1-yl}ethoxy)ethan-1-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide