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2-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}-1,2-oxazinane
(4aS,7aR)-N-cyclopentyl-4-[(dimethylcarbamoyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(1-{1-[(2-methoxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
2-(3-hydroxypropanoyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[3-(furan-2-yl)propyl]piperidin-4-amine
5-(3-methoxyphenoxymethyl)-N-methyl-N-(piperidin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-(2-cyclopentylacetyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N,N-dimethyl-1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-amine
4-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
8-[2-(dimethylamino)benzoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-(4-methylphenyl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]urea
N-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
6,6-dimethyl-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-5-oxothiomorpholine-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)pyrrolidine-1-carboxamide
7-{2-[2-(propan-2-yl)-1H-1,3-benzodiazol-1-yl]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
1-(6-methylpyridin-2-yl)-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
3-hydroxy-3-({[(2-hydroxypyridin-3-yl)methyl]amino}methyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
methyl 3-(but-2-ynoyl)-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N,N-dimethyl-4-[(1E)-3-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)prop-1-en-1-yl]aniline
7-(2-hydroxyethyl)-2-[1-(2-methylphenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[1-(1H-imidazol-1-yl)butan-2-yl]urea
2-methoxy-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]phenol
1-[4-(2,5-dimethylphenyl)piperazin-1-yl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-{2-[methyl(phenyl)amino]ethyl}-3-(piperidin-3-yl)benzamide
4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-(oxan-4-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-benzyl-5-(cyclopentylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
6-[(6-hydroxy-1,4-oxazepan-6-yl)methyl]-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methoxy}phenyl)acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methyl-2-oxopentanamide
(4-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholin-2-yl)methanamine
2-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
N-[2-(oxolan-2-ylmethoxy)phenyl]-4-phenylpiperidine-1-carboxamide
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine
methyl N-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}carbamate
(2S,3S)-2-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]-3-methylpentanamide
3-{[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[(3S,4R)-1-(benzenesulfonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(2S,4R)-4-(cyclooctylamino)-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-benzoyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-amine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethylpyrrolidin-2-yl)methyl]-5-methoxybenzamide
9-(6-methylpyridazin-3-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol