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4-{2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-(3-tert-butyl-5-methylphenyl)-2-fluorobenzamide
1-cyclopropyl-N-[(4-fluorophenyl)methyl]-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-(2-methoxyethyl)-2-methyl-7-(piperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(4-fluorophenyl)methyl]-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-(azetidine-1-carbonyl)-1-(2-methoxyphenyl)-1H-pyrazole
2-[2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]-1H-imidazole
(3S,4S)-1-[2-(1,1-dioxo-1λ6-thian-4-yl)acetyl]-4-propylpyrrolidine-3-carboxylic acid
(3R,4S)-4-cyclopropyl-1-(4-fluoro-2-methylbenzoyl)pyrrolidin-3-amine
2-{9-[(3-methoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
8-{[2-(trifluoromethoxy)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
3-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1-(2-oxopiperidin-3-yl)urea
4-[(2,2-dimethyloxan-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(4-methyl-3-phenylpiperazine-1-carbonyl)pyrazin-2-ol
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
butyl 3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carboxylate
3-(1H-indol-3-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
3-(methylsulfamoyl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
(4aS,8aR)-6-(furan-2-carbonyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1-butyl-5-(cyclohex-3-en-1-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
(1s,4s)-4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]-5,6-dimethyl-1H-1,3-benzodiazole
2-phenyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
(2S,4R)-4-amino-N-ethyl-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidine-2-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(2-phenylethyl)piperidin-1-yl]propan-1-one
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(thiophen-3-yl)acetamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
2-phenyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)azetidine
1-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
(3R,5S)-N-[2-(dimethylamino)ethyl]-1-(2-methylpropyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
(3aS,6aS)-2-(furan-3-ylmethyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[1'-(2-fluorobenzoyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
4-[2-(2-fluorophenyl)ethyl]-3-[(4-methylpiperazin-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-methoxypropyl)-2,3-dihydro-1H-indene-2-carboxamide
2-cyclopropyl-6-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-4-oxo-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-chloro-4-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]phenol
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[2-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](methyl)amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
(4aS,8aR)-6-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]pyridin-2-amine
1-[5-(2-methyl-1,3-benzothiazol-5-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
N-(4-phenylbutyl)-1,9-dioxaspiro[5.5]undecan-4-amine
3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[(1-hydroxycyclohexyl)methyl]urea
N-[1-(furan-2-carbonyl)piperidin-4-yl]-3-phenyl-1H-pyrazole-4-carboxamide