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1-[1-(5-methoxy-4-oxo-1,4-dihydropyridine-2-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
(2S,4S)-4-amino-1-[(2,5-dimethoxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
1-[3-methoxy-5-(trifluoromethyl)phenyl]-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrrole-2-carboxamide
{4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4-oxazepan-6-yl}methanol
3-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}amino)-2-methoxypyridine-3-carbonitrile
2-[(3-methoxyphenyl)amino]-N-[2-(N-methylmethanesulfonamido)ethyl]butanamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1,3-thiazole-4-carboxamide
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(azocan-1-yl)propan-1-one
3-(2-methoxyphenyl)-6-[4-(pyrrolidin-1-yl)piperidin-1-yl]pyridazine
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(4-fluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(dimethylamino)benzamide
3-[(3R,4S)-4-(dimethylamino)-1-[(4-fluoro-2-methylphenyl)methyl]piperidin-3-yl]propan-1-ol
N-(2-{4-[(2,3-dimethyl-1H-indol-7-yl)methyl]morpholin-2-yl}ethyl)acetamide
4-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
3-(2-oxopyrrolidin-1-yl)-N-[phenyl(pyridin-4-yl)methyl]propanamide
3-hexyl-8-(1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-[4-(thiophen-2-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
8-methyl-5-{4-[1-(1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]pyridin-2-yl}quinoline
3-[(3R,4S)-1-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N-[2-(1H-imidazol-1-yl)propyl]-2,6-dimethylquinoline-4-carboxamide
1-[1-(3-cyclopentylpropyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
2-[4-(oxane-4-carbonyl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(prop-2-en-1-yl)acetamide
2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
N-methyl-5-[(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
2-ethoxy-6-({3-[(4-fluorophenyl)amino]piperidin-1-yl}methyl)phenol
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,4-triazole
8-(3-hydroxypropanoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
(3S,4R)-4-(3-fluorophenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(2,6-difluoro-3-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
3-benzyl-4-[2-(2-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(pyridin-3-yl)-7-[2-(1H-pyrrol-1-yl)pentanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2,3-dimethylquinoxaline-6-carboxamide
N-{[4-(hydroxymethyl)phenyl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methylpentan-1-one
2-chloro-N-{2-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
4-(3-{[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]oxy}benzoyl)morpholine
3-{5-[2-(diethylamino)ethyl]-1,3,4-thiadiazol-2-yl}-1-[(1-methyl-5-oxopyrrolidin-3-yl)methyl]urea
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
(3R,4S)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3,4-dimethylpiperidin-4-ol