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(1S,6R)-9-(1,3-thiazol-2-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methyl-6-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidin-4-ol
2-[3,5-dimethyl-4-(2,3,6-trimethylquinoline-4-amido)-1H-pyrazol-1-yl]acetic acid
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-chloro-6-fluorophenyl)acetamide
2-methoxy-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}acetamide
1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-6-(thian-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-ethyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]urea
1-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-yl}-4-phenylpiperazine
5-fluoro-3-methyl-2-{[4-(1-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-indole
ethyl 1-[(4-acetamidophenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(2-methylpropanoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
(1S,6R)-9-{[5-(hydroxymethyl)furan-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
(5S,9aS,9bS)-5-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{[2-(methylamino)pyrimidin-5-yl]formamido}-N-phenylpropanamide
(2R,3R)-1'-(pyrazin-2-yl)-3-(1,2,3,6-tetrahydropyridin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(2,3-dihydroxypropyl)-6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N2-{3-[(2-ethylphenyl)carbamoyl]phenyl}pyrrolidine-1,2-dicarboxamide
(2S,4S)-4-amino-N-ethyl-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
(3S,4S)-1-(morpholine-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
ethyl 1-[3-({[(2-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperidine-3-carboxylate
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(2-phenylethyl)azepan-4-amine
(3R)-3,4,4-trimethyl-1-(2-methylpyrimidin-4-yl)pyrrolidin-3-ol
(1R,5R)-3-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
2-(4-{[(2S,5R)-5-{[ethyl(methyl)amino]methyl}oxolan-2-yl]methyl}phenoxy)-N-methylacetamide
2-methyl-5-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-ethyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}butanamide
1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-imidazole-5-carboxamide
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]butan-1-one
1-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-3-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]urea
N-[(1R,3R)-3-aminocyclopentyl]-1-ethyl-1H-pyrazole-4-sulfonamide
methyl 4-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)thiophene-2-carboxylate
2-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]-N,N-bis(propan-2-yl)benzamide
6-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyrazine-2-carboxamide
5-[(dimethylamino)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
(2R,3R)-1'-(1H-imidazol-2-ylmethyl)-3-(4-methylpiperazin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
7-(3-methoxypyrazin-2-yl)-2-methyl-N-(oxolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-ethyl-N-phenyl-3-[4-(pyrazin-2-yl)piperazin-1-yl]propanamide
(3S,9R)-11-(2-methoxybenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-{5-[2-(dimethylamino)-4-methylpyrimidin-5-yl]-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-methyl-5-{[2-methyl-2-(morpholin-4-yl)propyl]amino}-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-phenoxybutyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-benzyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one