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(1S,5R)-3-benzoyl-N,N-diethyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-({4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)ethyl]acetamide
2,6-dimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
2-cyclobutyl-5-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,3,4-oxadiazole
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
2-[4-(4,4-difluoropiperidin-1-yl)-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
5-(2,3-difluoro-6-methoxyphenyl)-1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[4-(2-cyanophenyl)-8-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]cyclopentanecarboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-2-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-N-(thiophen-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-ethyl-1-methyl-3-[1-(6-phenylpyridazin-3-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-benzyl-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-methanesulfonyl-N-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-amine
3-methyl-3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[4-(trifluoromethoxy)phenyl]urea
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
(4aS,7aR)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(1,4-dioxan-2-ylmethyl)-3-[(2,2,2-trifluoroethyl)sulfamoyl]benzamide
2-ethyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-cyclopropyl-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine-2-carboxamide
(2S,4R)-N-ethyl-4-(3-hydroxy-4-methylbenzamido)-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
2-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}acetamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)piperidine
5-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3S,4S)-3-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]-4-hydroxypyrrolidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine-3-carboxylate
cyclopentyl 4-({[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)benzoate
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-[(2E)-3-phenylprop-2-en-1-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(2-ethoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-1-[4-(1,3-thiazol-4-yl)phenyl]urea
bis(1,3-oxazol-4-ylmethyl)({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amine
2-oxo-N-phenyl-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetamide
7-(4-methoxy-3-methylbenzenesulfonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2-fluorophenyl)-4-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-[(1-cyclopentanecarbonylpiperidin-4-yl)formamido]-3-(1H-imidazol-4-yl)propanoic acid
{4-[4-(5-methylfuran-2-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
7-(propan-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
3-(2-{2-methyl-4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,3-diazinane-2,4-dione
2-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-imidazole
N-(dimethyl-1,2-oxazol-4-yl)-2-(3-fluorophenyl)-3-oxopiperazine-1-carboxamide
(2E)-3-(1,3-benzothiazol-2-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)prop-2-enamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(4-hydroxyphenyl)benzamide
(4aR,7aS)-1-ethyl-4-(8-fluoroquinoline-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,3,4-trimethoxybenzamide
1-[1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
7-(methylsulfanyl)-3-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-[({5-[1-(6-cyclopropylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol