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4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-6-methyl-1-(2-methylphenyl)piperazin-2-one
N,N-diethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-(8-methoxyquinolin-5-yl)-6-(propan-2-yloxy)pyrimidin-2-amine
methyl 8-{[3-(furan-2-yl)phenyl]methyl}-1-[(3-methoxyphenyl)methoxy]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(3aR,7aS)-2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
(1R,5S)-N-(6-methoxyquinolin-8-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3R,9aR)-3-benzyl-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2,3,6-trimethylquinoline-4-carbonyl)piperidine-2-carboxylic acid
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,6,6-trimethyl-5-oxothiomorpholine-3-carboxamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(quinolin-5-ylmethyl)amine
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-{4-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenyl}-N-methylmethanesulfonamide
(1R,7S)-6-(4-methyl-3-oxopiperazine-1-carbonyl)-3-(2-phenoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-amine
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-(pyridin-2-yl)pyrimidine
2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methylpyrimidine-5-carboxamide
2-[2-(ethoxymethyl)pyrimidin-5-yl]-N,N,3,6-tetramethylquinoline-4-carboxamide
3-[(4aR,7aS)-4-[(4-fluoro-2-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
4-{[(1R)-2-hydroxy-1-phenylethyl]sulfamoyl}-N-(propan-2-yl)benzamide
(1-{[1-(3-methylbenzenesulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-cyclohexyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-amine
N-[(2-methoxyphenyl)methyl]-2-{methyl[1-(pyrimidin-4-yl)ethyl]amino}acetamide
N,N-dimethyl-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-2-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3,4-dimethoxyphenyl)methyl]-5-(1H-pyrrol-2-yl)-1,2,4-oxadiazole
2-(cyclopentylmethyl)-1-[2-(dimethylamino)ethyl]-N,6-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}ethyl]methylamine
7-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(2-fluorophenoxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
N-(1H-imidazol-2-ylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,2,3,4-tetrahydronaphthalen-2-yl)imidazo[1,2-a]pyridine-6-carboxamide
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrazine
2-methyl-4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}quinoline
1-(1H-pyrrole-3-carbonyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
3-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-1-(4-phenylphenyl)urea
1-(4-{methyl[1-(2-phenylethyl)piperidin-3-yl]amino}piperidin-1-yl)ethan-1-one
2,6-dioxo-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1S,6R)-9-[5-(methoxymethyl)thiophene-2-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
4-{methyl[2-(oxan-4-yl)ethyl]sulfamoyl}-N-propylbenzamide
1-({5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
3-hydroxy-N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-(2-methylphenyl)pyrrolidine-1-carboxamide
1-ethyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[5-(6-methylhept-5-en-2-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-5-ethyl-N-propyl-1,2-oxazole-3-carboxamide