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(3aS,6aS)-2-cyclobutanecarbonyl-5-(2-methyl-6-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-N-(propan-2-yl)propanamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]-3-(1-methylpiperidin-4-yl)propanamide
1,6-dimethyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-methyl-1,2-oxazole-5-carboxamide
5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
N-methyl-5-{[(oxolan-3-yl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[4-(8-methoxyquinolin-5-yl)phenyl]ethan-1-ol
[(5-{1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(1R,5R)-6-[(3,5-dimethoxyphenyl)methyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
8-(2,4-dimethylpyrimidine-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
[(3R,4R)-1-[(3-ethoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(1S,5R)-3-(quinolin-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-4,6-dimethyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydropyridin-2-one
2-methyl-N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-phenylpiperazine-1-carboxamide
5-(3-chloro-5-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(oxan-4-yl)propanamide
1-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)carbamoyl]methyl}piperidine-4-carboxamide
[(3-methoxyphenyl)methyl](methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N6-(3-methoxypropyl)-N5-methyl-N5-(2,2,6,6-tetramethylpiperidin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
2-{1-[(2-methylphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-benzyl-8-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
7-(cyclopropylmethyl)-2-{[4-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
2-propyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
6-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]-2,3-dimethylquinoxaline
1-(2-methylpropyl)-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
(1,4-dioxan-2-ylmethyl)(methyl)[(3-methylphenyl)methyl]amine
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-propylpyridine-4-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-fluorobenzene-1-sulfonamide
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N,2,6,8-tetramethylquinoline-4-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-propylpropanamide
4-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)-2,3-dihydro-1H-imidazol-2-one
2-methyl-8-{[3-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
propyl N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
2-benzyl-9-[(2R)-2-hydroxy-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2-ethoxybenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
9-[2-(2,3-difluorophenyl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-benzoyl-N-methyl-N-[(3-methylthiophen-2-yl)methyl]piperidin-4-amine
3-[2-(2-fluorophenyl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-(3-methylphenyl)piperidine-1-carboxamide