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1-(4-methanesulfonylpiperazin-1-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[(2-methoxyphenyl)methyl]-N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4-phenyl-1H-pyrazol-5-amine
1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1H-indazole
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{4-[(propan-2-yl)carbamoyl]pyridin-2-yl}-decahydro-2,7-naphthyridine-2-carboxamide
1-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)-3,5-dimethyl-1H-pyrazole
2,2-dimethyl-3-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-{[4-(benzyloxy)phenyl]methyl}-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(4-methyl-1,3-thiazol-5-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)propanamide
(2S,4S,5R)-4-[4-(hydroxymethyl)piperidine-1-carbonyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
2-(4-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylpropyl)amino]methyl}piperidin-2-one
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(3-methylbut-2-en-1-yl)-8-(pyridine-3-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
4-(2-methyl-1H-imidazol-1-yl)-1-[4-(4-methylphenoxy)piperidin-1-yl]butan-1-one
4-[(1S,2R)-2-{2-[2-(ethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}-1-hydroxypropyl]phenol
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-methyl-N-(pyridin-3-ylmethyl)propanamide
2,5-dimethyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1,3-thiazole-4-carboxamide
3-{[ethyl(oxolan-2-ylmethyl)amino]methyl}-N-(pyrazin-2-yl)benzamide
N-{2-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]ethyl}aniline
5-(2-chlorophenyl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]furan-2-carboxamide
9-methoxy-7-(3-methoxyphenyl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-(4,5-dimethylfuran-2-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(3-methylphenoxy)azetidine
4-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-1-methylpiperazin-2-one
ethyl 1-[2-(dimethylamino)ethyl]-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-4-(pyridine-3-carbonyl)-1,4-diazepan-2-one
4-[5-(aminomethyl)pyridin-2-yl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 4-(5-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-[2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamido]-N-[(3-methylphenyl)methyl]benzamide
N-methyl-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
methyl 3-{[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]carbamoyl}propanoate
3-(4-chlorophenyl)-5-(cyclopropylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3S,4S)-4-(4-fluorophenyl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-ol
4-methyl-2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-ethyl-5-(piperidin-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(3R,4S)-3,4-dimethyl-1-(5-{[(4-methylphenyl)sulfanyl]methyl}furan-2-carbonyl)piperidin-4-ol
2-(1H-1,3-benzodiazol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-cyano-N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]benzene-1-sulfonamide
1-(4-{[2-hydroxy-5-(6-methoxypyridin-2-yl)phenyl]methyl}piperazin-1-yl)ethan-1-one
methyl 6-(2,2-dimethylpropanoyl)-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S)-1-[3-(2-methoxyethyl)-1-propyl-1H-1,2,4-triazol-5-yl]-2-phenylethan-1-ol
N-[5-({cyclohexyl[2-(ethylsulfanyl)ethyl]carbamoyl}amino)-2-fluorophenyl]acetamide
1-[5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-phenylazepane