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4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(quinolin-8-ylmethyl)piperidin-4-ol
(1S,5R)-6-(4-fluoro-2-methylbenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-{1-[(4-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}benzonitrile
1-(3-methoxyphenyl)-4-{2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetyl}piperazin-2-one
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
1-ethyl-4-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,2-dihydropyridin-2-one
(4aR,8aS)-N,N-dimethyl-1-(2,3,4-trifluorobenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
(3R,7S,8aS)-7-{[(2,5-dimethylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(4-fluorophenoxymethyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1,3-oxazole-4-carboxamide
{3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-5-methyl-1,2-oxazol-4-yl}methanol
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazine-1-sulfonamide
1-(2-methoxyphenyl)-4-[3-(piperidin-1-yl)propanoyl]piperazin-2-one
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[2-(5-methylfuran-2-yl)ethyl]piperidin-4-amine
2-methyl-1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
1-(1-oxo-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-2-yl)pyrrolidin-2-one
(3aR,5R,6S,7aS)-2-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
[(3R,4R)-1-(4-tert-butylbenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
4-({4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-(propan-2-yl)pyrimidine
2-{8-cyclopentyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carboxylic acid
N-ethyl-5-({4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)pyrimidin-2-amine
4-[(4-ethoxyphenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
7-methoxy-4-methyl-2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]quinazoline
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-methyl-2-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
methyl 4-{[4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carbonyl]amino}-3-methylbenzoate
2-{1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}-1,3-benzothiazole
4-[(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-2-yl)methyl]morpholine
3-(2-oxopyrrolidin-1-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
N-[(2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)oxane-2-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-(4-methoxypiperidin-1-yl)pyridine-3-carboxamide
3-ethyl-1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidine-3-carboxylic acid
(1R,5R)-3-(1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(2S,6S)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-phenylethan-1-one
4-[(benzyloxy)methyl]-1-[(dimethyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole
5-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[(3R,4R)-4-(hydroxymethyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
N-(2-fluorophenyl)-3-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
N-{[3-(cyclopentyloxy)-4-methoxyphenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
3-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-4H-1,2,4-triazole
1-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-[5-(4-methylphenyl)furan-2-yl]propan-1-one
N-[(4-phenyloxan-4-yl)methyl]-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
2-methoxy-3-[4-(pyrrolidin-1-ylmethyl)phenyl]pyridine
1-(methoxymethyl)-N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}cyclobutane-1-carboxamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one