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N-ethyl-6-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-N-methylpyridine-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-({[3-(benzyloxy)phenyl]carbamoyl}(methyl)amino)-N-methylbutanamide
(3S,4S)-1-(6-methylpyridine-2-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(3S,4R)-3-(dimethylamino)-N-ethyl-4-(4-methylphenyl)pyrrolidine-1-carboxamide
2,5,7-trimethyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]quinoline-4-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-imidazol-1-yl)butan-1-one
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[3-(thiophen-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methoxypyrimidine-5-carboxamide
6-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1,4-oxazepan-6-ol
8-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,3-dimethoxyphenyl)-2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}acetic acid
2-methyl-4-(3-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}phenyl)butan-2-ol
(2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(piperidin-1-yl)butanamide
5-ethyl-2-methyl-4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyrimidine
4-(4-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}butyl)morpholine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2,3-dimethyl-1H-indole-5-carboxamide
5-[2-(difluoromethoxy)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-(2-phenylpropan-2-yl)pyrrolidine-3-carboxamide
ethyl 1-(1H-indole-5-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
N'-cyclooctyl-N-[4-(pyridin-2-yl)butyl]butanediamide
N-(2-methanesulfonylethyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)furan-2-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(pyridin-4-ylsulfanyl)acetamide
2-[(dimethyl-1,3-thiazol-5-yl)methyl]-7-(3-methylbenzoyl)-2,7-diazaspiro[4.5]decane
1-({4-[(1E)-pent-1-en-1-yl]thiophen-2-yl}methyl)piperazine
1-[(2-fluoro-4-methoxyphenyl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
N-({5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}cyclopropanamine
1-(2-methylpyridin-4-yl)-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
(3S)-1-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)piperidine-3-carboxylic acid
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
5-{[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole
7-[4-(1-ethoxyethyl)phenyl]-1,2-dihydroisoquinolin-1-one
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-cyclopropyl-1-(4-methanesulfonylphenyl)-5-(5-propyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(isoquinolin-5-ylmethyl)piperidin-3-amine
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(2-methoxyethyl)-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
N-[(2-methoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4,4-difluoro-N-(2-methyl-1-benzofuran-7-yl)piperidine-1-carboxamide
1-[1-(1-methylpiperidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
(2S,4R)-N-ethyl-4-[(3E)-hex-3-enamido]-1-(1-methyl-1H-imidazole-5-carbonyl)pyrrolidine-2-carboxamide