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N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]piperidin-2-one
N,N,4-trimethyl-3-{[methyl(pentan-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-cyclohexyl-N-cyclopropyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
[2-ethoxy-5-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]methanol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
(1R,6S)-9-methyl-3-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-3,9-diazabicyclo[4.2.1]nonane
1-(4-benzylpiperazin-1-yl)-3-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]propan-1-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine-4-carboxamide
1-methyl-N-[2-(morpholin-4-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(2-hydroxyethoxy)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(1,3-thiazol-2-ylmethyl)amine
3-({5-[4-(1,2,3-thiadiazol-4-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
1-(2-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)pyrrolidin-2-one
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]benzonitrile
5-(2-ethylpiperidine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
5-hydroxy-N-methyl-N-(2-phenoxyethyl)pyrazine-2-carboxamide
2-(2-hydroxyphenoxy)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
3-methyl-7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
methyl 5-[(2,2-dimethyloxan-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
5-[(5-acetylthiophen-3-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
9-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-{1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-(oxolan-2-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-[(3R,4S)-1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-(2,5-dimethoxyphenyl)-4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
(4aS,8aR)-1-butyl-6-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-decahydro-1,6-naphthyridin-2-one
5-[2-(3-fluorophenyl)piperidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
{9-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-(cyclopropylmethyl)-5-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)-1,2,4-triazin-3-amine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
(3aS,7aR)-2-(2-chloro-4,5-difluorobenzoyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(4-fluorophenyl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]cyclopropane-1-carboxamide
[7-(1H-pyrazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-{[1-(dimethylsulfamoyl)pyrrolidin-3-yl]methyl}benzamide
1-(2-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(3aS,6aS)-2-methyl-5-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)(quinoxalin-2-ylmethyl)amine
3-(2-phenoxyethyl)-8-(1-propyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2S,4S)-N-ethyl-4-(2-hydroxy-5-methylbenzamido)-1-(3-methoxypropyl)pyrrolidine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]cyclohexanecarboxamide
3-[(2R,3R,6R)-5-[(2-ethylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-methyl-2-(methylamino)-1,3-thiazole-5-carboxamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}acetamide